European Journal of Medicinal Chemistry

, том 46 , издание 3 , страницы 819-824

Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships

潘斌 Pan Bin ^{1, 2, 3}

Renzheng Huang ⁴

Likang Zheng ^{1, 2, 3}

Chen Chen ^{1, 2, 3}

Shiqing Han ^{1, 2, 3}

Di Qu ⁴

Mingli Zhu ^{1, 2, 3}

Ping Wei ^{1, 2, 3}

Скрыть аффилиации авторов Показать аффилиации авторов: 4 аффилиации

College of Biotechnology and Pharmaceutical Engineering

Nanjing University of technology |

Nanjing 210009 China |

⁴

Key Laboratory of Medical Molecular Virology of Ministry of Education and Ministry of Pulic Health, Institute of Medical Microbiology and Institutes of Biomedical Sciences, Shanghai Medical School of Fudan University Box 228, Shanghai 200032, China |

Тип публикации: Journal Article

Дата публикации: 2011-03-01

Elsevier

European Journal of Medicinal Chemistry

scimago Q1

wos Q1

БС1

SJR: 1.142

CiteScore: 11.3

Impact factor: 5.9

ISSN: 02235234, 17683254

DOI: 10.1016/j.ejmech.2010.12.014

Скопировать DOI

PubMed ID: 21255878

Organic Chemistry

Drug Discovery

General Medicine

Pharmacology

Краткое описание

Rational designed novel thiazolidiones were synthesized and evaluated for antibiofilm activity. The active derivatives were not only potent inhibitors of Staphylococcus epidermidis biofilm growth but also efficient antibacterial agents. 3f showed 4-fold higher activity (6.25 μM) in the biofilms dispersal assay and significantly higher antibacterial activity (MIC 3.125 μM) in comparison to the 3-(5-((6- (ethoxycarbonyl)-5-(benzo[1,3]dioxol-5-yl)-3-oxo-7-phenyl- thiazolo[3,2-a]pyrimidin-2(5H)-ylidene)methyl)furan-2-yl)benzoic acid (1).

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1 цитирование

Шетнев Антон

к.х.н.

79 публикаций, 767 цитирований

Индекс Хирша: 15

Московский физико-технический институт

Ярославский государственный медицинский университет

Ярославский государственный педагогический университет имени К. Д. Ушинского

1 цитирование

Нефедова Анна

12 публикаций, 50 цитирований

Индекс Хирша: 4

Институт органической и физической химии им. А.Е. Арбузова КазНЦ РАН

Области научных интересов

Кристаллохимия

Органическая химия

Супрамолекулярная химия

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Pan Bin 潘. 斌. et al. Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships // European Journal of Medicinal Chemistry. 2011. Vol. 46. No. 3. pp. 819-824.

ГОСТ со всеми авторами (до 50) Скопировать

Pan Bin 潘. 斌., Huang R., Zheng L., Chen C., Han S., Qu D., Zhu M., Wei P. Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships // European Journal of Medicinal Chemistry. 2011. Vol. 46. No. 3. pp. 819-824.

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TY - JOUR

DO - 10.1016/j.ejmech.2010.12.014

UR - https://doi.org/10.1016/j.ejmech.2010.12.014

TI - Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships

T2 - European Journal of Medicinal Chemistry

AU - Pan Bin, 潘斌

AU - Huang, Renzheng

AU - Zheng, Likang

AU - Chen, Chen

AU - Han, Shiqing

AU - Qu, Di

AU - Zhu, Mingli

AU - Wei, Ping

PY - 2011

DA - 2011/03/01

PB - Elsevier

SP - 819-824

IS - 3

VL - 46

PMID - 21255878

SN - 0223-5234

SN - 1768-3254

ER -

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@article{2011_Pan Bin,

author = {潘斌 Pan Bin and Renzheng Huang and Likang Zheng and Chen Chen and Shiqing Han and Di Qu and Mingli Zhu and Ping Wei},

title = {Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships},

journal = {European Journal of Medicinal Chemistry},

year = {2011},

volume = {46},

publisher = {Elsevier},

month = {mar},

url = {https://doi.org/10.1016/j.ejmech.2010.12.014},

number = {3},

pages = {819--824},

doi = {10.1016/j.ejmech.2010.12.014}

}

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MLA Скопировать

Pan Bin, 潘. 斌., et al. “Thiazolidione derivatives as novel antibiofilm agents: Design, synthesis, biological evaluation, and structure–activity relationships.” European Journal of Medicinal Chemistry, vol. 46, no. 3, Mar. 2011, pp. 819-824. https://doi.org/10.1016/j.ejmech.2010.12.014.

Издатель

Elsevier

Журнал

European Journal of Medicinal Chemistry

scimago Q1

wos Q1

БС1

SJR

1.142

CiteScore

11.3

Impact factor

5.9

ISSN

02235234 (Print)

17683254 (Electronic)

Профили

Хан