volume 366 issue 10 pages 2252-2256

Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines

Yannan Zhu 1
He Zhao 1
Qiuyun Li 1
Fang Bo 2
Yi-ning Wang 1
Gang Qi 1
1
 
Faculty of Chemistry and Chemical Engineering Yancheng Institute of Technology Yancheng 224051 People's Republic of China
2
 
Yancheng Tongwei Solar Energy Co., Ltd Yancheng 224000 People's Republic of China
Publication typeJournal Article
Publication date2024-04-24
scimago Q1
wos Q1
SJR0.930
CiteScore8.0
Impact factor4.0
ISSN16154150, 16154169
General Chemistry
Abstract

The domino annulation reactions of o‐aminotrifluoroacetophenone derivatives and MBH carbonates enabled by PPh3 have been reported, which provide a series of tetrahydrofuro[3,2‐b]indolines containing a CF3‐substituted tetrasubstituted carbon stereocenters in yields of 74 to 95% and >20:1 dr. In this process, MBH carbonates were used as C1/C3 synthons. The MTT assay shows that the products exhibit the activity of inhibitory effect on proliferation on Hela cancer cell line.

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Zhu Y. et al. Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines // Advanced Synthesis and Catalysis. 2024. Vol. 366. No. 10. pp. 2252-2256.
GOST all authors (up to 50) Copy
Zhu Y., Zhao H., Li Q., Fang Bo, Wang Y., Qi G. Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines // Advanced Synthesis and Catalysis. 2024. Vol. 366. No. 10. pp. 2252-2256.
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TY - JOUR
DO - 10.1002/adsc.202400205
UR - https://onlinelibrary.wiley.com/doi/10.1002/adsc.202400205
TI - Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines
T2 - Advanced Synthesis and Catalysis
AU - Zhu, Yannan
AU - Zhao, He
AU - Li, Qiuyun
AU - Fang Bo
AU - Wang, Yi-ning
AU - Qi, Gang
PY - 2024
DA - 2024/04/24
PB - Wiley
SP - 2252-2256
IS - 10
VL - 366
SN - 1615-4150
SN - 1615-4169
ER -
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BibTex (up to 50 authors) Copy
@article{2024_Zhu,
author = {Yannan Zhu and He Zhao and Qiuyun Li and Fang Bo and Yi-ning Wang and Gang Qi},
title = {Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines},
journal = {Advanced Synthesis and Catalysis},
year = {2024},
volume = {366},
publisher = {Wiley},
month = {apr},
url = {https://onlinelibrary.wiley.com/doi/10.1002/adsc.202400205},
number = {10},
pages = {2252--2256},
doi = {10.1002/adsc.202400205}
}
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Zhu, Yannan, et al. “Phosphine‐Catalyzed Domino Annulation Reactions of o‐Aminotrifluoroacetophenone Derivatives with Morita−Baylis−Hillman Carbonates: Construction of Tetrahydrofuro[3,2‐b]indolines.” Advanced Synthesis and Catalysis, vol. 366, no. 10, Apr. 2024, pp. 2252-2256. https://onlinelibrary.wiley.com/doi/10.1002/adsc.202400205.