volume 7 issue 5 pages 226-230

The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification

G R Bourne 1
S. R. Moss 1
P. J. PHILLIPS 1
B Shuker 1
1
 
Safety of Medicines Department, ICI Pharmaceuticals Division, Alderley Park, Nr Macclesfield, Cheshire SK10 4TG, UK
Publication typeJournal Article
Publication date1980-05-01
scimago Q3
wos Q2
SJR0.427
CiteScore4.0
Impact factor2.0
ISSN10765174, 10969888
Biochemistry
Spectroscopy
Molecular Medicine
Abstract
The metabolic fate of the synthetic prostaglandin cloprostenol ('Estrumate') in the cow has been studied. Following intramuscular administration of 0.5 mg and 10 mg of [14C]cloprostenol to cows urinary excretion accounted for 58.2% and 56.3% of the dose respectively. Unchanged cloprostenol and its tetranor acid, probably formed by beta-oxidation, were the major components identified in urine. The tetranor acid was also present as a glucuronide conjugate. This synthetic prostaglandin analogue is apparently a poor substrate for the enzymes 15-hydroxyprostaglandin dehydrogenase and 13,14-reductase, which are responsible for the rapid metabolic deactivation of endogenous prostaglandins, as no components identified in urine were found to have undergone metabolic attack at the C-15 atom in the cloprostenol molecule.
Found 
Found 

Top-30

Journals

1
2
3
4
Journal of Dairy Science
4 publications, 28.57%
Chemico-Biological Interactions
1 publication, 7.14%
Theriogenology
1 publication, 7.14%
Journal of Clinical Pharmacology
1 publication, 7.14%
Journal für praktische Chemie
1 publication, 7.14%
Journal of Veterinary Pharmacology and Therapeutics
1 publication, 7.14%
Reproduction in Domestic Animals
1 publication, 7.14%
Drug Metabolism Reviews
1 publication, 7.14%
1
2
3
4

Publishers

1
2
3
4
5
6
Elsevier
6 publications, 42.86%
Wiley
4 publications, 28.57%
Taylor & Francis
1 publication, 7.14%
1
2
3
4
5
6
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
14
Share
Cite this
GOST |
Cite this
GOST Copy
Bourne G. R. et al. The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification // Journal of Mass Spectrometry. 1980. Vol. 7. No. 5. pp. 226-230.
GOST all authors (up to 50) Copy
Bourne G. R., Moss S. R., PHILLIPS P. J., Shuker B. The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification // Journal of Mass Spectrometry. 1980. Vol. 7. No. 5. pp. 226-230.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1002/bms.1200070509
UR - https://doi.org/10.1002/bms.1200070509
TI - The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification
T2 - Journal of Mass Spectrometry
AU - Bourne, G R
AU - Moss, S. R.
AU - PHILLIPS, P. J.
AU - Shuker, B
PY - 1980
DA - 1980/05/01
PB - Wiley
SP - 226-230
IS - 5
VL - 7
PMID - 7417700
SN - 1076-5174
SN - 1096-9888
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{1980_Bourne,
author = {G R Bourne and S. R. Moss and P. J. PHILLIPS and B Shuker},
title = {The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification},
journal = {Journal of Mass Spectrometry},
year = {1980},
volume = {7},
publisher = {Wiley},
month = {may},
url = {https://doi.org/10.1002/bms.1200070509},
number = {5},
pages = {226--230},
doi = {10.1002/bms.1200070509}
}
MLA
Cite this
MLA Copy
Bourne, G. R., et al. “The metabolic fate of the synthetic prostaglandin cloprostenol (‘Estrumate’) in the cow: Use of ion cluster techniques to facilitate metabolite identification.” Journal of Mass Spectrometry, vol. 7, no. 5, May. 1980, pp. 226-230. https://doi.org/10.1002/bms.1200070509.