том 24 издание 15 страницы 3721-3724

Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones

Тип публикацииJournal Article
Дата публикации2018-02-19
SCImago Q1
WOS Q2
БС1
SJR0.803
CiteScore5.8
Impact factor3.6
ISSN09476539, 15213765
General Chemistry
Catalysis
Organic Chemistry
Краткое описание
An intramolecular catalytic dearomatization of phenols via gold carbene species proceeded to provide 2-azaspiro[4.5]decan-3-ones. The use of NHC ligand and water as a co-solvent was critical for achieving high reactivity. This reaction did not require hazardous diazo compounds as carbene sources and proceeded even under air. The obtained spirocyclic product could be readily transformed into a gabapentin derivative by hydrogenation and deprotection.
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ГОСТ |
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Ito M. et al. Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones // Chemistry - A European Journal. 2018. Vol. 24. No. 15. pp. 3721-3724.
ГОСТ со всеми авторами (до 50) Скопировать
Ito M., KAWASAKI R., Kanyiva K. S., Shibata T. Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones // Chemistry - A European Journal. 2018. Vol. 24. No. 15. pp. 3721-3724.
RIS |
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TY - JOUR
DO - 10.1002/chem.201800314
UR - https://doi.org/10.1002/chem.201800314
TI - Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones
T2 - Chemistry - A European Journal
AU - Ito, Mitsuo
AU - KAWASAKI, Ryosuke
AU - Kanyiva, Kyalo Stephen
AU - Shibata, Takanori
PY - 2018
DA - 2018/02/19
PB - Wiley
SP - 3721-3724
IS - 15
VL - 24
PMID - 29372752
SN - 0947-6539
SN - 1521-3765
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2018_Ito,
author = {Mitsuo Ito and Ryosuke KAWASAKI and Kyalo Stephen Kanyiva and Takanori Shibata},
title = {Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones},
journal = {Chemistry - A European Journal},
year = {2018},
volume = {24},
publisher = {Wiley},
month = {feb},
url = {https://doi.org/10.1002/chem.201800314},
number = {15},
pages = {3721--3724},
doi = {10.1002/chem.201800314}
}
MLA
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Ito, Mitsuo, et al. “Catalytic Dearomative Spirocyclization via Gold Carbene Species Derived from Ynamides: Efficient Synthesis of 2-Azaspiro[4.5]decan-3-ones.” Chemistry - A European Journal, vol. 24, no. 15, Feb. 2018, pp. 3721-3724. https://doi.org/10.1002/chem.201800314.
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