C3‐Functionalization of Imidazo[1,2‐a]pyridines
Among nitrogen‐containing organic compounds, imidazo[1,2‐a]pyridines, and especially C3‐functionalized imidazo[1,2‐a]pyridines, have a wide range of industrial applications in the fields of optics, material science, and organometallics. This scaffolds also have various medicinal uses due to their antiviral, cytotoxic, antibacterial, fungicidal, and antiinflammatory activities as they are found in many commercially available drugs such as Alpidem, Miroprofen, and Zolimidine. In this review, we summarized and classified the latest synthetic methods for the preparation of C3‐functionalized imidazo[1,2‐a]pyridines based on the type of the substituents on the 3‐position of imidazo[1,2‐a]pyridine including C3‐alkylation, C3‐arylation, C3‐carbonylation, C3‐sulfenylation, C3‐selenation, C3‐N‐Substitution, C3‐phosphonation, and C3‐halogenation.
Top-30
Journals
|
2
4
6
8
10
12
14
|
|
|
Journal of Organic Chemistry
13 publications, 12.38%
|
|
|
Advanced Synthesis and Catalysis
7 publications, 6.67%
|
|
|
European Journal of Organic Chemistry
6 publications, 5.71%
|
|
|
Asian Journal of Organic Chemistry
6 publications, 5.71%
|
|
|
Tetrahedron Letters
5 publications, 4.76%
|
|
|
Organic and Biomolecular Chemistry
5 publications, 4.76%
|
|
|
ChemistrySelect
4 publications, 3.81%
|
|
|
New Journal of Chemistry
4 publications, 3.81%
|
|
|
Organic Letters
3 publications, 2.86%
|
|
|
Chinese Journal of Organic Chemistry
3 publications, 2.86%
|
|
|
Tetrahedron
3 publications, 2.86%
|
|
|
Green Chemistry
3 publications, 2.86%
|
|
|
RSC Advances
3 publications, 2.86%
|
|
|
Beilstein Journal of Organic Chemistry
2 publications, 1.9%
|
|
|
Molecules
2 publications, 1.9%
|
|
|
Molecular Diversity
2 publications, 1.9%
|
|
|
ACS Omega
2 publications, 1.9%
|
|
|
Organic Chemistry Frontiers
2 publications, 1.9%
|
|
|
Synthetic Communications
2 publications, 1.9%
|
|
|
Synthesis
2 publications, 1.9%
|
|
|
Heterocycles
2 publications, 1.9%
|
|
|
Letters in Organic Chemistry
2 publications, 1.9%
|
|
|
Russian Journal of Organic Chemistry
1 publication, 0.95%
|
|
|
Current Organic Chemistry
1 publication, 0.95%
|
|
|
Current Chemical Biology
1 publication, 0.95%
|
|
|
Catalysts
1 publication, 0.95%
|
|
|
MolBank
1 publication, 0.95%
|
|
|
Pharmaceuticals
1 publication, 0.95%
|
|
|
Medicinal Chemistry Research
1 publication, 0.95%
|
|
|
Green Synthesis and Catalysis
1 publication, 0.95%
|
|
|
2
4
6
8
10
12
14
|
Publishers
|
5
10
15
20
25
30
|
|
|
Wiley
27 publications, 25.71%
|
|
|
American Chemical Society (ACS)
18 publications, 17.14%
|
|
|
Royal Society of Chemistry (RSC)
18 publications, 17.14%
|
|
|
Elsevier
12 publications, 11.43%
|
|
|
Springer Nature
6 publications, 5.71%
|
|
|
MDPI
5 publications, 4.76%
|
|
|
Bentham Science Publishers Ltd.
4 publications, 3.81%
|
|
|
Shanghai Institute of Organic Chemistry
3 publications, 2.86%
|
|
|
Georg Thieme Verlag KG
3 publications, 2.86%
|
|
|
Beilstein-Institut
2 publications, 1.9%
|
|
|
Taylor & Francis
2 publications, 1.9%
|
|
|
The Japan Institute of Heterocyclic Chemistry
2 publications, 1.9%
|
|
|
Pleiades Publishing
1 publication, 0.95%
|
|
|
Korean Society of Industrial Engineering Chemistry
1 publication, 0.95%
|
|
|
Asian Journal of Chemistry
1 publication, 0.95%
|
|
|
5
10
15
20
25
30
|
- We do not take into account publications without a DOI.
- Statistics recalculated weekly.