Design, Synthesis, and Biological Evaluation of New Territrem B Analogues
Тип публикации: Journal Article
Дата публикации: 2005-04-18
scimago Q3
wos Q3
БС2
SJR: 0.425
CiteScore: 3.5
Impact factor: 2.5
ISSN: 16121872, 16121880
PubMed ID:
17192004
General Chemistry
Biochemistry
Molecular Biology
General Medicine
Molecular Medicine
Bioengineering
Краткое описание
Some 23 analogues of the potent acetylcholinesterase (AChE) inhibitor territrem B (1) were designed, synthesized, and tested for their biological activities. Some of the new synthetic derivatives exhibited IC50 values for AChE inhibition in the upper micromolar range. Molecular-modeling studies indicated that a planar conformation seems to be crucial for AChE inhibition. The two N-atoms of the piperazine moieties in 5o, 5p, and 5r might further enhance the inhibitory effects. The cytotoxicities of selected compounds against six human tumor cell lines were also determined.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Для доступа к списку цитирований публикации необходимо авторизоваться.
Топ-30
Журналы
|
1
|
|
|
Bioorganic and Medicinal Chemistry Letters
1 публикация, 11.11%
|
|
|
Mendeleev Communications
1 публикация, 11.11%
|
|
|
Journal of Medicinal Chemistry
1 публикация, 11.11%
|
|
|
ACS Medicinal Chemistry Letters
1 публикация, 11.11%
|
|
|
Studies in Natural Products Chemistry
1 публикация, 11.11%
|
|
|
Journal of Pharmacy and Pharmacology
1 публикация, 11.11%
|
|
|
Asian Journal of Poultry Science
1 публикация, 11.11%
|
|
|
Asian Journal of Animal Sciences
1 публикация, 11.11%
|
|
|
1
|
Издатели
|
1
2
3
|
|
|
Elsevier
3 публикации, 33.33%
|
|
|
American Chemical Society (ACS)
2 публикации, 22.22%
|
|
|
Science Alert
2 публикации, 22.22%
|
|
|
Wiley
1 публикация, 11.11%
|
|
|
1
2
3
|
- Мы не учитываем публикации, у которых нет DOI.
- Статистика публикаций обновляется еженедельно.
Вы ученый?
Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Метрики
9
Всего цитирований:
9
Цитирований c 2025:
0
Цитировать
ГОСТ |
RIS |
BibTex |
MLA
Цитировать
ГОСТ
Скопировать
Jiang X. et al. Design, Synthesis, and Biological Evaluation of New Territrem B Analogues // Chemistry and Biodiversity. 2005. Vol. 2. No. 4. pp. 557-567.
ГОСТ со всеми авторами (до 50)
Скопировать
Jiang X., Ao L., Zhou C., Yang L., Zhang Q., Li H., Sun L., Wu X., Bai H., Zhou Y. Design, Synthesis, and Biological Evaluation of New Territrem B Analogues // Chemistry and Biodiversity. 2005. Vol. 2. No. 4. pp. 557-567.
Цитировать
RIS
Скопировать
TY - JOUR
DO - 10.1002/cbdv.200590036
UR - https://doi.org/10.1002/cbdv.200590036
TI - Design, Synthesis, and Biological Evaluation of New Territrem B Analogues
T2 - Chemistry and Biodiversity
AU - Jiang, Xiangrui
AU - Ao, Lei
AU - Zhou, Changxin
AU - Yang, Leixiang
AU - Zhang, Qijun
AU - Li, Haibo
AU - Sun, Lian-li
AU - Wu, Xiumei
AU - Bai, Hua
AU - Zhou, Yu-Tao
PY - 2005
DA - 2005/04/18
PB - Wiley
SP - 557-567
IS - 4
VL - 2
PMID - 17192004
SN - 1612-1872
SN - 1612-1880
ER -
Цитировать
BibTex (до 50 авторов)
Скопировать
@article{2005_Jiang,
author = {Xiangrui Jiang and Lei Ao and Changxin Zhou and Leixiang Yang and Qijun Zhang and Haibo Li and Lian-li Sun and Xiumei Wu and Hua Bai and Yu-Tao Zhou},
title = {Design, Synthesis, and Biological Evaluation of New Territrem B Analogues},
journal = {Chemistry and Biodiversity},
year = {2005},
volume = {2},
publisher = {Wiley},
month = {apr},
url = {https://doi.org/10.1002/cbdv.200590036},
number = {4},
pages = {557--567},
doi = {10.1002/cbdv.200590036}
}
Цитировать
MLA
Скопировать
Jiang, Xiangrui, et al. “Design, Synthesis, and Biological Evaluation of New Territrem B Analogues.” Chemistry and Biodiversity, vol. 2, no. 4, Apr. 2005, pp. 557-567. https://doi.org/10.1002/cbdv.200590036.