том 34 издание 5 страницы 1511-1517

Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones

Тип публикацииJournal Article
Дата публикации1997-09-01
scimago Q3
wos Q2
БС2
SJR0.362
CiteScore4.7
Impact factor2.4
ISSN0022152X, 19435193
Organic Chemistry
Краткое описание
Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates 1a,b react with het-eroarylamines 2 to give alkyl 2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-heteroarylaminopropenoates 3-13. These were cyclized into fused 3-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-4H-azolo- (or azino)-pyrim-idin-4-ones 14-18. 2-Benzoyl-2-ethoxycarbonyl-1-ethenyl group can be easily removed from 3-(2-benzoyl-2-ethoxycarbonyl-1-emenyl)amino-8-memyl-4H-pyrido[1,2-a]pyrimidin-4-one (14) to give 3-amino-8-methyl-4H-pyrido[1,2-a]pyrimidin-4-one (19). The structure of 1a was confirmed by X-ray analysis.
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Journal of Heterocyclic Chemistry
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ГОСТ |
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Strah S. et al. Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones // Journal of Heterocyclic Chemistry. 1997. Vol. 34. No. 5. pp. 1511-1517.
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Strah S., Golobič A., Golic L., Stanovnik B. Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones // Journal of Heterocyclic Chemistry. 1997. Vol. 34. No. 5. pp. 1511-1517.
RIS |
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TY - JOUR
DO - 10.1002/jhet.5570340521
UR - https://doi.org/10.1002/jhet.5570340521
TI - Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones
T2 - Journal of Heterocyclic Chemistry
AU - Strah, Sonja
AU - Golobič, Amalija
AU - Golic, Ljubo
AU - Stanovnik, Branko
PY - 1997
DA - 1997/09/01
PB - Wiley
SP - 1511-1517
IS - 5
VL - 34
SN - 0022-152X
SN - 1943-5193
ER -
BibTex |
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@article{1997_Strah,
author = {Sonja Strah and Amalija Golobič and Ljubo Golic and Branko Stanovnik},
title = {Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones},
journal = {Journal of Heterocyclic Chemistry},
year = {1997},
volume = {34},
publisher = {Wiley},
month = {sep},
url = {https://doi.org/10.1002/jhet.5570340521},
number = {5},
pages = {1511--1517},
doi = {10.1002/jhet.5570340521}
}
MLA
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Strah, Sonja, et al. “Alkyl (E,Z)-2-(2-benzoyl-2-ethoxycarbonyl-1-ethenyl)amino-3-dimethylaminopropenoates in the synthesis of fused pyrimidinones. A facile route to 3-aminoazino-4H-pyrimidin-4-ones.” Journal of Heterocyclic Chemistry, vol. 34, no. 5, Sep. 1997, pp. 1511-1517. https://doi.org/10.1002/jhet.5570340521.