том 43 издание 4 страницы 1031-1035

Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction

Тип публикацииJournal Article
Дата публикации2006-07-01
scimago Q3
wos Q2
БС2
SJR0.362
CiteScore4.7
Impact factor2.4
ISSN0022152X, 19435193
Organic Chemistry
Краткое описание
Efficient syntheses of dibenz[b,f][1,4]oxazepin-11(10H)-one, 5,10-dihydro-11H-dibenzo[b,e][1,4]-diazepin-11-one and 5,11-dihydro-6H-dibenz[b,e]azepin-6-one are described using a tandem reductionlactamization sequence. Precursors for these ring systems are available in 1-3 steps using nucleophilic aromatic substitution and Ullmann coupling methodology. Direct reduction-lactamization of these compounds using iron powder in acetic acid at 115° affords the target heterocycles in ≥90% yield.
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ГОСТ |
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Bunce R. A., Schammerhorn J. E. Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction // Journal of Heterocyclic Chemistry. 2006. Vol. 43. No. 4. pp. 1031-1035.
ГОСТ со всеми авторами (до 50) Скопировать
Bunce R. A., Schammerhorn J. E. Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction // Journal of Heterocyclic Chemistry. 2006. Vol. 43. No. 4. pp. 1031-1035.
RIS |
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TY - JOUR
DO - 10.1002/jhet.5570430432
UR - https://doi.org/10.1002/jhet.5570430432
TI - Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction
T2 - Journal of Heterocyclic Chemistry
AU - Bunce, Richard A
AU - Schammerhorn, James E
PY - 2006
DA - 2006/07/01
PB - Wiley
SP - 1031-1035
IS - 4
VL - 43
SN - 0022-152X
SN - 1943-5193
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2006_Bunce,
author = {Richard A Bunce and James E Schammerhorn},
title = {Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction},
journal = {Journal of Heterocyclic Chemistry},
year = {2006},
volume = {43},
publisher = {Wiley},
month = {jul},
url = {https://doi.org/10.1002/jhet.5570430432},
number = {4},
pages = {1031--1035},
doi = {10.1002/jhet.5570430432}
}
MLA
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Bunce, Richard A., and James E Schammerhorn. “Dibenzo-fused seven-membered nitrogen heterocycles by a tandem reduction-lactamization reaction.” Journal of Heterocyclic Chemistry, vol. 43, no. 4, Jul. 2006, pp. 1031-1035. https://doi.org/10.1002/jhet.5570430432.