volume 52 issue 5 pages 303-308

Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde

Konstantin F Suzdalev 1
Natalia I Vikrischuk 1
Kseniya A Prikhodko 1
Elena Yu Shasheva 1
Sergey V. Kurbatov 1
Saida K Bogus 2
Pavel A Galenko Yaroshevsky 2
Publication typeJournal Article
Publication date2016-05-01
scimago Q4
wos Q4
SJR0.243
CiteScore2.7
Impact factor1.0
ISSN00093122, 15738353
Organic Chemistry
Abstract
A two-step approach towards the synthesis of imidazo[1,2-a]indoles from 2-chloroindole-3-carbaldehyde has been developed. It comprises the N-alkylation of indole ring by 2-bromo-1,1-diethoxyethane followed by a treatment with aromatic amine hydrochlorides. The reaction proceeds as a nucleophilic substitution of the chlorine atom at position 2 of the indole ring followed by cyclization along with the condensation at the aldehyde group. Imidazo[1,2-a]indoles were isolated as protonated Schiff bases. Their structure was proved by 1H and 13C NMR spectroscopy and X-ray structural analysis.
Found 
Found 

Top-30

Journals

1
2
3
Russian Journal of General Chemistry
3 publications, 42.86%
Tetrahedron Letters
1 publication, 14.29%
ChemInform
1 publication, 14.29%
Mendeleev Communications
1 publication, 14.29%
Journal of Heterocyclic Chemistry
1 publication, 14.29%
1
2
3

Publishers

1
2
3
Pleiades Publishing
3 publications, 42.86%
Wiley
2 publications, 28.57%
Elsevier
1 publication, 14.29%
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 publication, 14.29%
1
2
3
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
7
Share
Cite this
GOST |
Cite this
GOST Copy
Suzdalev K. F. et al. Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde // Chemistry of Heterocyclic Compounds. 2016. Vol. 52. No. 5. pp. 303-308.
GOST all authors (up to 50) Copy
Suzdalev K. F., Vikrischuk N. I., Prikhodko K. A., Shasheva E. Yu., Kurbatov S. V., Bogus S. K., Galenko Yaroshevsky P. A. Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde // Chemistry of Heterocyclic Compounds. 2016. Vol. 52. No. 5. pp. 303-308.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1007/s10593-016-1882-y
UR - https://doi.org/10.1007/s10593-016-1882-y
TI - Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde
T2 - Chemistry of Heterocyclic Compounds
AU - Suzdalev, Konstantin F
AU - Vikrischuk, Natalia I
AU - Prikhodko, Kseniya A
AU - Shasheva, Elena Yu
AU - Kurbatov, Sergey V.
AU - Bogus, Saida K
AU - Galenko Yaroshevsky, Pavel A
PY - 2016
DA - 2016/05/01
PB - Springer Nature
SP - 303-308
IS - 5
VL - 52
SN - 0009-3122
SN - 1573-8353
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2016_Suzdalev,
author = {Konstantin F Suzdalev and Natalia I Vikrischuk and Kseniya A Prikhodko and Elena Yu Shasheva and Sergey V. Kurbatov and Saida K Bogus and Pavel A Galenko Yaroshevsky},
title = {Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde},
journal = {Chemistry of Heterocyclic Compounds},
year = {2016},
volume = {52},
publisher = {Springer Nature},
month = {may},
url = {https://doi.org/10.1007/s10593-016-1882-y},
number = {5},
pages = {303--308},
doi = {10.1007/s10593-016-1882-y}
}
MLA
Cite this
MLA Copy
Suzdalev, Konstantin F., et al. “Synthesis of Imidazo[1,2-a]Indoles from 2-Chloroindole-3-Carbaldehyde.” Chemistry of Heterocyclic Compounds, vol. 52, no. 5, May. 2016, pp. 303-308. https://doi.org/10.1007/s10593-016-1882-y.