volume 57 issue 4 pages 448-454

Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines

Vladimir А Ostrovskii 1
Gevorg G Danagulyan 2, 3
Olga M. Nesterova 1
Yulia N Pavlyukova 1
Vladimir V Tolstyakov 1
Olga S Zarubina 1
Pavel А Slepukhin 4
Yana L Esaulkova 5
Anna А Muryleva 5
Vladimir V. Zarubaev 5
Rostislav E. Trifonov 1
Publication typeJournal Article
Publication date2021-04-01
scimago Q4
wos Q4
SJR0.243
CiteScore2.7
Impact factor1.0
ISSN00093122, 15738353
Organic Chemistry
Abstract
Nonannulated tetrazolylpyrimidines in the structure of which the heterocyclic fragments are separated by hydrazinocarbonylmethyl, methylpyrazolyl groups or a sulfur atom were synthesized. Some of these compounds showed moderate in vitro activity against H1N1 subtype of influenza A virus. The selectivity index of the anti-influenza action of {5-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1H-tetrazol-1-yl}acetic acid, which has very low cytotoxicity, was twice as high as the selectivity index of the reference drug rimantadine.
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Ostrovskii V. А. et al. Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines // Chemistry of Heterocyclic Compounds. 2021. Vol. 57. No. 4. pp. 448-454.
GOST all authors (up to 50) Copy
Ostrovskii V. А., Danagulyan G. G., Nesterova O. M., Pavlyukova Y. N., Tolstyakov V. V., Zarubina O. S., Slepukhin P. А., Esaulkova Y. L., Muryleva A. А., Zarubaev V. V., Trifonov R. E. Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines // Chemistry of Heterocyclic Compounds. 2021. Vol. 57. No. 4. pp. 448-454.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1007/s10593-021-02922-6
UR - https://doi.org/10.1007/s10593-021-02922-6
TI - Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines
T2 - Chemistry of Heterocyclic Compounds
AU - Ostrovskii, Vladimir А
AU - Danagulyan, Gevorg G
AU - Nesterova, Olga M.
AU - Pavlyukova, Yulia N
AU - Tolstyakov, Vladimir V
AU - Zarubina, Olga S
AU - Slepukhin, Pavel А
AU - Esaulkova, Yana L
AU - Muryleva, Anna А
AU - Zarubaev, Vladimir V.
AU - Trifonov, Rostislav E.
PY - 2021
DA - 2021/04/01
PB - Springer Nature
SP - 448-454
IS - 4
VL - 57
PMID - 34007083
SN - 0009-3122
SN - 1573-8353
ER -
BibTex |
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BibTex (up to 50 authors) Copy
@article{2021_Ostrovskii,
author = {Vladimir А Ostrovskii and Gevorg G Danagulyan and Olga M. Nesterova and Yulia N Pavlyukova and Vladimir V Tolstyakov and Olga S Zarubina and Pavel А Slepukhin and Yana L Esaulkova and Anna А Muryleva and Vladimir V. Zarubaev and Rostislav E. Trifonov},
title = {Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines},
journal = {Chemistry of Heterocyclic Compounds},
year = {2021},
volume = {57},
publisher = {Springer Nature},
month = {apr},
url = {https://doi.org/10.1007/s10593-021-02922-6},
number = {4},
pages = {448--454},
doi = {10.1007/s10593-021-02922-6}
}
MLA
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MLA Copy
Ostrovskii, Vladimir А., et al. “Synthesis and antiviral activity of nonannulated tetrazolylpyrimidines.” Chemistry of Heterocyclic Compounds, vol. 57, no. 4, Apr. 2021, pp. 448-454. https://doi.org/10.1007/s10593-021-02922-6.