volume 125 issue 1 pages 129-139

Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents

Shiv Kumar 1
Nitin Kumar 2
Sushma Drabu 3
Md Akram Minhaj 1
1
 
Division of Pharmaceutical Chemistry, Department of Pharmacy, IEC College of Engineering and Technology, Greater Noida, India
2
 
Department of Pharmaceutical Technology, Meerut Institute of Engineering and Technology, Meerut, India
3
 
Maharaja Surajmal Institute of Pharmacy, Janak Puri, India
Publication typeJournal Article
Publication date2013-01-01
scimago Q3
wos Q3
SJR0.315
CiteScore3.0
Impact factor2.0
ISSN09743626, 09737103, 02534134
General Chemistry
Abstract
Twelve compounds belonging to series N-[3-chloro-2-oxo-4-(substituted)phenylazetidin-1-yl]-2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide (5a–l) were synthesized. These compounds were evaluated for their in vitro antibacterial against E. coli, S. aureus, K. pneumoniae, P. aeruginosa and antifungal activity against C. albicans, A. niger and A. flavus by cup-plate method. Structures of all the newly synthesized compounds were confirmed by their spectral data interpretation. Compound 5g having p-dimethylaminophenyl group on 4-position of azetidinone ring attached to N-atom of acetamido group on 1-position of 3-methyl-1H-quinoxaline-2-one, was found to be active against all the bacterial and fungal strains under investigation.
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GOST Copy
Kumar S. et al. Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents // Journal of Chemical Sciences. 2013. Vol. 125. No. 1. pp. 129-139.
GOST all authors (up to 50) Copy
Kumar S., Kumar N., Drabu S., Minhaj M. A. Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents // Journal of Chemical Sciences. 2013. Vol. 125. No. 1. pp. 129-139.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1007/s12039-012-0354-x
UR - https://doi.org/10.1007/s12039-012-0354-x
TI - Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents
T2 - Journal of Chemical Sciences
AU - Kumar, Shiv
AU - Kumar, Nitin
AU - Drabu, Sushma
AU - Minhaj, Md Akram
PY - 2013
DA - 2013/01/01
PB - Springer Nature
SP - 129-139
IS - 1
VL - 125
SN - 0974-3626
SN - 0973-7103
SN - 0253-4134
ER -
BibTex |
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BibTex (up to 50 authors) Copy
@article{2013_Kumar,
author = {Shiv Kumar and Nitin Kumar and Sushma Drabu and Md Akram Minhaj},
title = {Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents},
journal = {Journal of Chemical Sciences},
year = {2013},
volume = {125},
publisher = {Springer Nature},
month = {jan},
url = {https://doi.org/10.1007/s12039-012-0354-x},
number = {1},
pages = {129--139},
doi = {10.1007/s12039-012-0354-x}
}
MLA
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MLA Copy
Kumar, Shiv, et al. “Synthesis of 2-(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetamide-based azetidinone derivatives as potent antibacterial and antifungal agents.” Journal of Chemical Sciences, vol. 125, no. 1, Jan. 2013, pp. 129-139. https://doi.org/10.1007/s12039-012-0354-x.