Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation
2
Microcare Laboratory, Surat, India
|
Publication type: Journal Article
Publication date: 2014-06-04
scimago Q2
wos Q3
SJR: 0.470
CiteScore: 5.1
Impact factor: 3.1
ISSN: 10542523, 15548120
Organic Chemistry
General Pharmacology, Toxicology and Pharmaceutics
Abstract
A new class of thiazolopyrimidine-based sulfonamides (5a–j) was synthesized from a parent compound 2-methoxy benzoic acid by multistep reaction in order to find new agents to fight against microbial infections. Substituted thiazolopyrimidines (3a–e) were prepared by cyclocondensation of substituted thiazolidinediones (2a–e) with urea in the presence of acid catalyst P2O5. Finally, desired compounds (5a–j) were synthesized from intermediates (4a–e) prepared from compounds (3a–e) by chlorosulfonation followed by condensation with corresponding benzothiazole moiety. The synthesized compounds were characterized by IR, 1H-NMR, 13C-NMR spectral data, and elemental analysis, and were evaluated for in vitro antimicrobial activity against certain bacterial and fungal strains using the broth microdilution method as well as antitubercular activity against H37Rv using Lowenstein–Jensen agar method.
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14
Total citations:
14
Citations from 2025:
1
(7.14%)
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Patel N. B., Purohit A. C., Rajani D. Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation // Medicinal Chemistry Research. 2014. Vol. 23. No. 11. pp. 4789-4802.
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Patel N. B., Purohit A. C., Rajani D. Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation // Medicinal Chemistry Research. 2014. Vol. 23. No. 11. pp. 4789-4802.
Cite this
RIS
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TY - JOUR
DO - 10.1007/s00044-014-1052-7
UR - https://doi.org/10.1007/s00044-014-1052-7
TI - Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation
T2 - Medicinal Chemistry Research
AU - Patel, Navin B
AU - Purohit, Amit C.
AU - Rajani, Dhanji
PY - 2014
DA - 2014/06/04
PB - Springer Nature
SP - 4789-4802
IS - 11
VL - 23
SN - 1054-2523
SN - 1554-8120
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2014_Patel,
author = {Navin B Patel and Amit C. Purohit and Dhanji Rajani},
title = {Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation},
journal = {Medicinal Chemistry Research},
year = {2014},
volume = {23},
publisher = {Springer Nature},
month = {jun},
url = {https://doi.org/10.1007/s00044-014-1052-7},
number = {11},
pages = {4789--4802},
doi = {10.1007/s00044-014-1052-7}
}
Cite this
MLA
Copy
Patel, Navin B., et al. “Newer thiazolopyrimidine-based sulfonamides clubbed with benzothiazole moiety: synthesis and biological evaluation.” Medicinal Chemistry Research, vol. 23, no. 11, Jun. 2014, pp. 4789-4802. https://doi.org/10.1007/s00044-014-1052-7.