Medicinal Chemistry Research

, volume 29 , issue 10 , pages 1751-1776

Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs

Sérgio Luiz Pinheiro ¹

Erick M C Pinheiro ²

Estela M.F. Muri ²

Jaqueline C Pessôa ¹

Mayara A Cadorini ³

Sandro J Greco ³

Hide authors affiliations Show authors affiliations: 3 affiliations

Instituto de Química, Universidade Federal Fluminense, Niterói, Brazil |

Departamento de Tecnologia Farmacêutica, Faculdade de Farmácia, Universidade Federal Fluminense, Niterói, Brazil |

Departamento de Química, Universidade Federal do Espírito Santo, Vitória, Brazil |

Publication type: Journal Article

Publication date: 2020-08-02

Springer Nature

Medicinal Chemistry Research

scimago Q2

wos Q3

SJR: 0.470

CiteScore: 5.1

Impact factor: 3.1

ISSN: 10542523, 15548120

DOI: 10.1007/s00044-020-02609-1

Copy DOI

Organic Chemistry

General Pharmacology, Toxicology and Pharmaceutics

Abstract

The [1,2,4]triazolo[1,5-a]pyrimidines (TPs) comprise an important class of non-naturally occurring small molecules that aroused the interest of researches. This scaffold is present in diverse important structures in agriculture and medicinal chemistry, such as antibacterial, antifungal, antiviral, antiparasitic, and anticancer. As over the decades the development of the chemistry and application of 1,2,4-triazolo[1,5-a]pyrimidines has continued and even accelerated, in this review, we thoroughly discussed the applications of TPs in both agriculture and medicinal chemistry highlighting the significance of this nucleus.

Found

2 citations

Babkov Denis

🤝

DSc in Pharmacy

78 publications, 827 citations, 60 reviews

h-index: 16

Volgograd State Medical University

1 citation

Sokolova Elena

20 publications, 245 citations

h-index: 10

Volgograd State Medical University

1 citation

Rasputin Nikolay

12 publications, 76 citations

h-index: 5

Postovsky Institute of Organic Synthesis of the Ural Branch of the Russian Academy of Sciences

Research interests

Heterocyclic compounds

Organic synthesis

Organometallic Chemistry

1 citation

Shchepochkin Alexandr

PhD in Chemistry

35 publications, 524 citations, 1 review

h-index: 13

Postovsky Institute of Organic Synthesis of the Ural Branch of the Russian Academy of Sciences

Ural Federal University

Research interests

"Smart" materials

Green chemistry

1 citation

Balyakin Ilya

🤝

PhD in Physics and Mathematics

31 publications, 352 citations, 17 reviews

h-index: 10

Institute of Metallurgy of the Ural Branch of the Russian Academy of Sciences

Ural Federal University

Harbin Institute of Technology

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GOST |

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GOST Copy

Pinheiro S. L. et al. Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs // Medicinal Chemistry Research. 2020. Vol. 29. No. 10. pp. 1751-1776.

GOST all authors (up to 50) Copy

Pinheiro S. L., Pinheiro E. M. C., Muri E. M., Pessôa J. C., Cadorini M. A., Greco S. J. Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs // Medicinal Chemistry Research. 2020. Vol. 29. No. 10. pp. 1751-1776.

RIS |

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RIS Copy

TY - JOUR

DO - 10.1007/s00044-020-02609-1

UR - https://link.springer.com/10.1007/s00044-020-02609-1

TI - Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs

T2 - Medicinal Chemistry Research

AU - Pinheiro, Sérgio Luiz

AU - Pinheiro, Erick M C

AU - Muri, Estela M.F.

AU - Pessôa, Jaqueline C

AU - Cadorini, Mayara A

AU - Greco, Sandro J

PY - 2020

DA - 2020/08/02

PB - Springer Nature

SP - 1751-1776

IS - 10

VL - 29

SN - 1054-2523

SN - 1554-8120

ER -

BibTex |

Cite this

BibTex (up to 50 authors) Copy

@article{2020_Pinheiro,

author = {Sérgio Luiz Pinheiro and Erick M C Pinheiro and Estela M.F. Muri and Jaqueline C Pessôa and Mayara A Cadorini and Sandro J Greco},

title = {Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs},

journal = {Medicinal Chemistry Research},

year = {2020},

volume = {29},

publisher = {Springer Nature},

month = {aug},

url = {https://link.springer.com/10.1007/s00044-020-02609-1},

number = {10},

pages = {1751--1776},

doi = {10.1007/s00044-020-02609-1}

}

MLA

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MLA Copy

Pinheiro, Sérgio Luiz, et al. “Biological activities of [1,2,4]triazolo[1,5-a]pyrimidines and analogs.” Medicinal Chemistry Research, vol. 29, no. 10, Aug. 2020, pp. 1751-1776. https://link.springer.com/10.1007/s00044-020-02609-1.

Publisher

Springer Nature

Journal

Medicinal Chemistry Research

scimago Q2

wos Q3

SJR

0.470

CiteScore

5.1

Impact factor

3.1

ISSN

10542523 (Print)

15548120 (Electronic)