volume 48 issue 4 pages 629-634

Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure

I P Tsypysheva 1
A V Kovalskaya 1
N S Makara 1
A N Lobov 1
I A Petrenko 1
E G Galkin 1
T A Sapozhnikova 1
F S Zarudii 1, 2
M. S. Yunusov 1
Publication typeJournal Article
Publication date2012-09-07
scimago Q3
wos Q4
SJR0.296
CiteScore1.3
Impact factor0.9
ISSN00093130, 15738388
General Chemistry
General Biochemistry, Genetics and Molecular Biology
Plant Science
Abstract
N-(methylcytisinyl)-N′-substituted ureas, N-substituted cytisine-12-carbamides, and cytisine-12-thiocarbamide were prepared by reaction of (–)-cytisine with urea and thiourea and of (–)-cytisine and its 12-N-methyl-3-amino derivative with isocyanates. Their specific nootropic activity was studied in vivo. The therapeutic index was determined for the lead compound. Promising candidates for further pharmacological testing were found.
Found 
Found 

Top-30

Journals

2
4
6
8
10
Chemistry of Natural Compounds
10 publications, 31.25%
Natural Product Research
4 publications, 12.5%
Pharmaceutical Chemistry Journal
2 publications, 6.25%
Journal of Agricultural and Food Chemistry
2 publications, 6.25%
Mini-Reviews in Medicinal Chemistry
1 publication, 3.13%
Chemical Papers
1 publication, 3.13%
European Journal of Medicinal Chemistry
1 publication, 3.13%
Tetrahedron Asymmetry
1 publication, 3.13%
Toxicology Reports
1 publication, 3.13%
Tetrahedron
1 publication, 3.13%
Journal of Photochemistry and Photobiology A: Chemistry
1 publication, 3.13%
Chemical Reviews
1 publication, 3.13%
Journal of Materials Chemistry A
1 publication, 3.13%
Russian Journal of Bioorganic Chemistry
1 publication, 3.13%
Journal of Structural Chemistry
1 publication, 3.13%
Russian Chemical Bulletin
1 publication, 3.13%
Mendeleev Communications
1 publication, 3.13%
Журнал Общей Химии
1 publication, 3.13%
2
4
6
8
10

Publishers

2
4
6
8
10
12
14
Springer Nature
14 publications, 43.75%
Elsevier
5 publications, 15.63%
Taylor & Francis
4 publications, 12.5%
American Chemical Society (ACS)
3 publications, 9.38%
Pleiades Publishing
2 publications, 6.25%
Bentham Science Publishers Ltd.
1 publication, 3.13%
Royal Society of Chemistry (RSC)
1 publication, 3.13%
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 publication, 3.13%
The Russian Academy of Sciences
1 publication, 3.13%
2
4
6
8
10
12
14
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
32
Share
Cite this
GOST |
Cite this
GOST Copy
Tsypysheva I. P. et al. Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure // Chemistry of Natural Compounds. 2012. Vol. 48. No. 4. pp. 629-634.
GOST all authors (up to 50) Copy
Tsypysheva I. P., Kovalskaya A. V., Makara N. S., Lobov A. N., Petrenko I. A., Galkin E. G., Sapozhnikova T. A., Zarudii F. S., Yunusov M. S. Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure // Chemistry of Natural Compounds. 2012. Vol. 48. No. 4. pp. 629-634.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1007/s10600-012-0329-7
UR - https://doi.org/10.1007/s10600-012-0329-7
TI - Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure
T2 - Chemistry of Natural Compounds
AU - Tsypysheva, I P
AU - Kovalskaya, A V
AU - Makara, N S
AU - Lobov, A N
AU - Petrenko, I A
AU - Galkin, E G
AU - Sapozhnikova, T A
AU - Zarudii, F S
AU - Yunusov, M. S.
PY - 2012
DA - 2012/09/07
PB - Springer Nature
SP - 629-634
IS - 4
VL - 48
SN - 0009-3130
SN - 1573-8388
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2012_Tsypysheva,
author = {I P Tsypysheva and A V Kovalskaya and N S Makara and A N Lobov and I A Petrenko and E G Galkin and T A Sapozhnikova and F S Zarudii and M. S. Yunusov},
title = {Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure},
journal = {Chemistry of Natural Compounds},
year = {2012},
volume = {48},
publisher = {Springer Nature},
month = {sep},
url = {https://doi.org/10.1007/s10600-012-0329-7},
number = {4},
pages = {629--634},
doi = {10.1007/s10600-012-0329-7}
}
MLA
Cite this
MLA Copy
Tsypysheva, I. P., et al. “Synthesis and specific nootropic activity of (–)-cytisine derivatives with carbamide and thiocarbamide moieties in their structure.” Chemistry of Natural Compounds, vol. 48, no. 4, Sep. 2012, pp. 629-634. https://doi.org/10.1007/s10600-012-0329-7.