Pharmaceutical Chemistry Journal

, том 51 , издание 7 , страницы 533-539

Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs

Тип публикации: Journal Article

Дата публикации: 2017-10-01

Springer Nature

Pharmaceutical Chemistry Journal

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SJR: 0.219

CiteScore: 1.4

Impact factor: 1

ISSN: 0091150X, 15739031

DOI: 10.1007/s11094-017-1649-5

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Drug Discovery

Pharmacology

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Thiazolo[2, 3-f]purine derivatives and their analogs – dihydrothiazolo[2, 3-f]purine, 7-(thietan-3-yl)purine, and 8-(2-hydroxypropylthio)purine derivatives – were synthesized. The compounds synthesized here had no effects on protein glycation reactions using glucose; they gave weak inhibition of glycogen phosphorylase; they had no hemorheological activity. Substances with hypotensive activity greater than that of Dibazol were found. A number of substances had hypoglycemic effects greater than those of chlorpropamide and Adebit. Two compounds inhibited dipeptidylpeptidase-4, but were less active than reference agent vildagliptin.

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Spasov A. et al. Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs // Pharmaceutical Chemistry Journal. 2017. Vol. 51. No. 7. pp. 533-539.

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Spasov A., Khaliullin F. A., Babkov D. A., Timirkhanova G. A., Kuznetsova V. A., Naumenko L. V., Muleeva D. R., Maika O. Yu., Prokhorova T. Yu., Sturova E. A. Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs // Pharmaceutical Chemistry Journal. 2017. Vol. 51. No. 7. pp. 533-539.

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TY - JOUR

DO - 10.1007/s11094-017-1649-5

UR - https://doi.org/10.1007/s11094-017-1649-5

TI - Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs

T2 - Pharmaceutical Chemistry Journal

AU - Spasov, A.A.

AU - Khaliullin, F A

AU - Babkov, D A

AU - Timirkhanova, G A

AU - Kuznetsova, V A

AU - Naumenko, L V

AU - Muleeva, D R

AU - Maika, O Yu

AU - Prokhorova, T Yu

AU - Sturova, E A

PY - 2017

DA - 2017/10/01

PB - Springer Nature

SP - 533-539

IS - 7

VL - 51

SN - 0091-150X

SN - 1573-9031

ER -

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@article{2017_Spasov,

author = {A.A. Spasov and F A Khaliullin and D A Babkov and G A Timirkhanova and V A Kuznetsova and L V Naumenko and D R Muleeva and O Yu Maika and T Yu Prokhorova and E A Sturova},

title = {Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs},

journal = {Pharmaceutical Chemistry Journal},

year = {2017},

volume = {51},

publisher = {Springer Nature},

month = {oct},

url = {https://doi.org/10.1007/s11094-017-1649-5},

number = {7},

pages = {533--539},

doi = {10.1007/s11094-017-1649-5}

}

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Spasov, A.A., et al. “Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs.” Pharmaceutical Chemistry Journal, vol. 51, no. 7, Oct. 2017, pp. 533-539. https://doi.org/10.1007/s11094-017-1649-5.