Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs
A.A. Spasov
1
,
F A Khaliullin
2
,
D A Babkov
1
,
G A Timirkhanova
2
,
V A Kuznetsova
1
,
L V Naumenko
1
,
D R Muleeva
1
,
O Yu Maika
1
,
T Yu Prokhorova
1
,
E A Sturova
1
Publication type: Journal Article
Publication date: 2017-10-01
scimago Q4
wos Q4
SJR: 0.219
CiteScore: 1.4
Impact factor: 1.0
ISSN: 0091150X, 15739031
Drug Discovery
Pharmacology
Abstract
Thiazolo[2, 3-f]purine derivatives and their analogs – dihydrothiazolo[2, 3-f]purine, 7-(thietan-3-yl)purine, and 8-(2-hydroxypropylthio)purine derivatives – were synthesized. The compounds synthesized here had no effects on protein glycation reactions using glucose; they gave weak inhibition of glycogen phosphorylase; they had no hemorheological activity. Substances with hypotensive activity greater than that of Dibazol were found. A number of substances had hypoglycemic effects greater than those of chlorpropamide and Adebit. Two compounds inhibited dipeptidylpeptidase-4, but were less active than reference agent vildagliptin.
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Total citations:
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Citations from 2024:
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Spasov A. et al. Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs // Pharmaceutical Chemistry Journal. 2017. Vol. 51. No. 7. pp. 533-539.
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Spasov A., Khaliullin F. A., Babkov D. A., Timirkhanova G. A., Kuznetsova V. A., Naumenko L. V., Muleeva D. R., Maika O. Yu., Prokhorova T. Yu., Sturova E. A. Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs // Pharmaceutical Chemistry Journal. 2017. Vol. 51. No. 7. pp. 533-539.
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RIS
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TY - JOUR
DO - 10.1007/s11094-017-1649-5
UR - https://doi.org/10.1007/s11094-017-1649-5
TI - Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs
T2 - Pharmaceutical Chemistry Journal
AU - Spasov, A.A.
AU - Khaliullin, F A
AU - Babkov, D A
AU - Timirkhanova, G A
AU - Kuznetsova, V A
AU - Naumenko, L V
AU - Muleeva, D R
AU - Maika, O Yu
AU - Prokhorova, T Yu
AU - Sturova, E A
PY - 2017
DA - 2017/10/01
PB - Springer Nature
SP - 533-539
IS - 7
VL - 51
SN - 0091-150X
SN - 1573-9031
ER -
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BibTex (up to 50 authors)
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@article{2017_Spasov,
author = {A.A. Spasov and F A Khaliullin and D A Babkov and G A Timirkhanova and V A Kuznetsova and L V Naumenko and D R Muleeva and O Yu Maika and T Yu Prokhorova and E A Sturova},
title = {Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs},
journal = {Pharmaceutical Chemistry Journal},
year = {2017},
volume = {51},
publisher = {Springer Nature},
month = {oct},
url = {https://doi.org/10.1007/s11094-017-1649-5},
number = {7},
pages = {533--539},
doi = {10.1007/s11094-017-1649-5}
}
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MLA
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Spasov, A.A., et al. “Synthesis and Antidiabetic Activity of Thiazolo[2,3-f]Purine Derivatives and Their Analogs.” Pharmaceutical Chemistry Journal, vol. 51, no. 7, Oct. 2017, pp. 533-539. https://doi.org/10.1007/s11094-017-1649-5.
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