Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections
A.S. Sokolova
1
,
D V Baranova
1, 2
,
O. I. Yarovaya
1, 2
,
D. S. Baev
1, 2
,
O A Polezhaeva
3
,
A V Zybkina
3
,
D. N. Shcherbakov
3
,
T G Tolstikova
1, 2
,
N. F. Salakhutdinov
1, 2
Publication type: Journal Article
Publication date: 2019-05-01
scimago Q3
SJR: 0.305
CiteScore: 2.8
Impact factor: —
ISSN: 10665285, 15739171
General Chemistry
Abstract
N-Heterocycle-containing (1S)-(+)-camphor-10-sulfonamide derivatives were synthesized. Their antiviral activity against the Ebola and Marburg viruses was estimated using a pseudovirus system based on the vesicular stomatitis virus. The derivatives bearing morpholine and triazole moieties demonstrated the highest inhibitory activity towards the Ebola virus glycoprotein. A moderate activity against the Marburg virus was found for a compound containing the piperidine moiety. A molecular modeling of the interaction between the synthesized derivatives and the binding site of glycoprotein of the Ebola virus was performed.
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Total citations:
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Citations from 2024:
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GOST
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Sokolova A. et al. Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections // Russian Chemical Bulletin. 2019. Vol. 68. No. 5. pp. 1041-1046.
GOST all authors (up to 50)
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Sokolova A., Baranova D. V., Yarovaya O. I., Baev D. S., Polezhaeva O. A., Zybkina A. V., Shcherbakov D. N., Tolstikova T. G., Salakhutdinov N. F. Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections // Russian Chemical Bulletin. 2019. Vol. 68. No. 5. pp. 1041-1046.
Cite this
RIS
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TY - JOUR
DO - 10.1007/s11172-019-2517-0
UR - https://doi.org/10.1007/s11172-019-2517-0
TI - Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections
T2 - Russian Chemical Bulletin
AU - Sokolova, A.S.
AU - Baranova, D V
AU - Yarovaya, O. I.
AU - Baev, D. S.
AU - Polezhaeva, O A
AU - Zybkina, A V
AU - Shcherbakov, D. N.
AU - Tolstikova, T G
AU - Salakhutdinov, N. F.
PY - 2019
DA - 2019/05/01
PB - Springer Nature
SP - 1041-1046
IS - 5
VL - 68
SN - 1066-5285
SN - 1573-9171
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2019_Sokolova,
author = {A.S. Sokolova and D V Baranova and O. I. Yarovaya and D. S. Baev and O A Polezhaeva and A V Zybkina and D. N. Shcherbakov and T G Tolstikova and N. F. Salakhutdinov},
title = {Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections},
journal = {Russian Chemical Bulletin},
year = {2019},
volume = {68},
publisher = {Springer Nature},
month = {may},
url = {https://doi.org/10.1007/s11172-019-2517-0},
number = {5},
pages = {1041--1046},
doi = {10.1007/s11172-019-2517-0}
}
Cite this
MLA
Copy
Sokolova, A.S., et al. “Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections.” Russian Chemical Bulletin, vol. 68, no. 5, May. 2019, pp. 1041-1046. https://doi.org/10.1007/s11172-019-2517-0.