volume 38 issue 7-8 pages 759-767

Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles

Publication typeJournal Article
Publication date2003-07-31
scimago Q1
wos Q1
SJR1.142
CiteScore11.3
Impact factor5.9
ISSN02235234, 17683254
Organic Chemistry
Drug Discovery
General Medicine
Pharmacology
Abstract
A series of 3-substituted 4-[5-(4-methoxy-2-nitrophenyl)-2-furfurylidene] amino-5-mercapto-1,2,4-triazoles (3) were synthesized. Aminomethylation of compounds 3 with formaldehyde and various secondary amines furnished Mannich bases 4 and 5. These compounds were characterized on the basis of IR, 1H-NMR, mass spectral data and elemental analysis. The newly synthesized compounds were screened for their anticancer activity against a panel of 60 cell lines derived from seven cancer types namely, lung, colon, melanoma, renal, ovarian, CNS and leukemia. Some of the compounds were slightly more potent.
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GOST |
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GOST Copy
Shivarama Holla B. et al. Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles // European Journal of Medicinal Chemistry. 2003. Vol. 38. No. 7-8. pp. 759-767.
GOST all authors (up to 50) Copy
Shivarama Holla B., Veerendra B., Shivananda M., Boja Poojary B. Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles // European Journal of Medicinal Chemistry. 2003. Vol. 38. No. 7-8. pp. 759-767.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1016/S0223-5234(03)00128-4
UR - https://doi.org/10.1016/S0223-5234(03)00128-4
TI - Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles
T2 - European Journal of Medicinal Chemistry
AU - Shivarama Holla, B.
AU - Veerendra, B.
AU - Shivananda, M.K.
AU - Boja Poojary, Boja
PY - 2003
DA - 2003/07/31
PB - Elsevier
SP - 759-767
IS - 7-8
VL - 38
PMID - 12932907
SN - 0223-5234
SN - 1768-3254
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2003_Shivarama Holla,
author = {B. Shivarama Holla and B. Veerendra and M.K. Shivananda and Boja Boja Poojary},
title = {Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles},
journal = {European Journal of Medicinal Chemistry},
year = {2003},
volume = {38},
publisher = {Elsevier},
month = {jul},
url = {https://doi.org/10.1016/S0223-5234(03)00128-4},
number = {7-8},
pages = {759--767},
doi = {10.1016/S0223-5234(03)00128-4}
}
MLA
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MLA Copy
Shivarama Holla, B., et al. “Synthesis characterization and anticancer activity studies on some Mannich bases derived from 1,2,4-triazoles.” European Journal of Medicinal Chemistry, vol. 38, no. 7-8, Jul. 2003, pp. 759-767. https://doi.org/10.1016/S0223-5234(03)00128-4.