volume 24 issue 1 pages 72-78

ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo

Henry Danahay 1
Clive McCarthy 2
Thomas Schofield 3
Tim Schofield 3
Roy Fox 4
Holly Charlton 4
Sarah Lilley 4
Juan Sabater 5
MATTHIAS SALATHÉ 6
Nathalie Baumlin 6
Stephen P Collingwood 2
Martin Gosling 2
1
 
Enterprise Therapeutics Ltd, 60 Science Park Square, Brighton BN1 9SB, UK. Electronic address: henry@enterprisetherapeutics.com.
2
 
Enterprise Therapeutics Ltd, 60 Science Park Square, Brighton BN1 9SB, UK.
3
 
Evotec UK Ltd, 114 Park Dr, Innovation Dr, Milton, Abingdon, OX14 4RZ, UK.
4
 
Sussex Drug Discovery Centre, School of Life Sciences, University of Sussex, Brighton, BN1 9RH, UK.
5
 
Department of Research, Mount Sinai Medical Center, 4300 Alton Rd, Miami Beach, FL 33140, USA.
Publication typeJournal Article
Publication date2025-01-01
scimago Q1
wos Q1
SJR1.772
CiteScore10.0
Impact factor6.0
ISSN15691993, 18735010
Abstract
Inhibiting ENaC in the airways of people with cystic fibrosis (pwCF) is hypothesized to enhance mucociliary clearance (MCC) and provide clinical benefit. Historically, inhaled ENaC blockers have failed to show benefit in pwCF challenging this hypothesis. It is however unknown whether the clinical doses were sufficient to provide the required long duration of action in the lungs and questions whether a novel candidate could offer advantages where others have failed?
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Danahay H. et al. ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo // Journal of Cystic Fibrosis. 2025. Vol. 24. No. 1. pp. 72-78.
GOST all authors (up to 50) Copy
Danahay H., McCarthy C., Schofield T., Schofield T., Fox R., Charlton H., Lilley S., Sabater J., SALATHÉ M., Baumlin N., Collingwood S. P., Gosling M. ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo // Journal of Cystic Fibrosis. 2025. Vol. 24. No. 1. pp. 72-78.
RIS |
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RIS Copy
TY - JOUR
DO - 10.1016/j.jcf.2024.06.002
UR - https://linkinghub.elsevier.com/retrieve/pii/S156919932400081X
TI - ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo
T2 - Journal of Cystic Fibrosis
AU - Danahay, Henry
AU - McCarthy, Clive
AU - Schofield, Thomas
AU - Schofield, Tim
AU - Fox, Roy
AU - Charlton, Holly
AU - Lilley, Sarah
AU - Sabater, Juan
AU - SALATHÉ, MATTHIAS
AU - Baumlin, Nathalie
AU - Collingwood, Stephen P
AU - Gosling, Martin
PY - 2025
DA - 2025/01/01
PB - Elsevier
SP - 72-78
IS - 1
VL - 24
PMID - 38851923
SN - 1569-1993
SN - 1873-5010
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2025_Danahay,
author = {Henry Danahay and Clive McCarthy and Thomas Schofield and Tim Schofield and Roy Fox and Holly Charlton and Sarah Lilley and Juan Sabater and MATTHIAS SALATHÉ and Nathalie Baumlin and Stephen P Collingwood and Martin Gosling},
title = {ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo},
journal = {Journal of Cystic Fibrosis},
year = {2025},
volume = {24},
publisher = {Elsevier},
month = {jan},
url = {https://linkinghub.elsevier.com/retrieve/pii/S156919932400081X},
number = {1},
pages = {72--78},
doi = {10.1016/j.jcf.2024.06.002}
}
MLA
Cite this
MLA Copy
Danahay, Henry, et al. “ETD001: A novel inhaled ENaC blocker with an extended duration of action in vivo.” Journal of Cystic Fibrosis, vol. 24, no. 1, Jan. 2025, pp. 72-78. https://linkinghub.elsevier.com/retrieve/pii/S156919932400081X.