volume 65 issue 41 pages 8461-8467

A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose

Publication typeJournal Article
Publication date2009-10-01
scimago Q3
wos Q2
SJR0.426
CiteScore4.1
Impact factor2.2
ISSN00404020, 14645416
Organic Chemistry
Drug Discovery
Biochemistry
Abstract
An enantioselective synthesis of suitably protected (1R,2S,4S,5S)-4-amino-1-(hydroxymethyl)bicyclo[3.1.0]hexan-2-ol, a key starting material for the synthesis of conformationally locked carbocyclic nucleosides, including the antiviral active North-methanocarba thymidine, is reported. Starting from 2-deoxyribose the target Boc-protected amine was prepared in 33% overall yield under condition that are ecologically friendlier than previous methods.
Found 
Found 

Top-30

Journals

1
2
Organic and Biomolecular Chemistry
2 publications, 10.53%
Journal of Antibiotics
1 publication, 5.26%
Coordination Chemistry Reviews
1 publication, 5.26%
Tetrahedron Asymmetry
1 publication, 5.26%
Tetrahedron Letters
1 publication, 5.26%
Bioorganic and Medicinal Chemistry
1 publication, 5.26%
International Journal of Quantum Chemistry
1 publication, 5.26%
Medicinal Research Reviews
1 publication, 5.26%
Chemistry - A European Journal
1 publication, 5.26%
Asian Journal of Organic Chemistry
1 publication, 5.26%
Organic Letters
1 publication, 5.26%
Journal of Organic Chemistry
1 publication, 5.26%
Crystal Growth and Design
1 publication, 5.26%
Chemical Society Reviews
1 publication, 5.26%
RSC Advances
1 publication, 5.26%
Synthesis
1 publication, 5.26%
International Journal of Molecular Sciences
1 publication, 5.26%
1
2

Publishers

1
2
3
4
5
Wiley
5 publications, 26.32%
Elsevier
4 publications, 21.05%
Royal Society of Chemistry (RSC)
4 publications, 21.05%
American Chemical Society (ACS)
3 publications, 15.79%
Springer Nature
1 publication, 5.26%
Georg Thieme Verlag KG
1 publication, 5.26%
MDPI
1 publication, 5.26%
1
2
3
4
5
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
19
Share
Cite this
GOST |
Cite this
GOST Copy
Ludek O. R., Marquez V. E. A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose // Tetrahedron. 2009. Vol. 65. No. 41. pp. 8461-8467.
GOST all authors (up to 50) Copy
Ludek O. R., Marquez V. E. A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose // Tetrahedron. 2009. Vol. 65. No. 41. pp. 8461-8467.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1016/j.tet.2009.08.035
UR - https://doi.org/10.1016/j.tet.2009.08.035
TI - A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose
T2 - Tetrahedron
AU - Ludek, Olaf R
AU - Marquez, Victor E.
PY - 2009
DA - 2009/10/01
PB - Elsevier
SP - 8461-8467
IS - 41
VL - 65
PMID - 20625519
SN - 0040-4020
SN - 1464-5416
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2009_Ludek,
author = {Olaf R Ludek and Victor E. Marquez},
title = {A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose},
journal = {Tetrahedron},
year = {2009},
volume = {65},
publisher = {Elsevier},
month = {oct},
url = {https://doi.org/10.1016/j.tet.2009.08.035},
number = {41},
pages = {8461--8467},
doi = {10.1016/j.tet.2009.08.035}
}
MLA
Cite this
MLA Copy
Ludek, Olaf R., and Victor E. Marquez. “A greener enantioselective synthesis of the antiviral agent North-methanocarbathymidine (N-MCT) from 2-deoxy-d-ribose.” Tetrahedron, vol. 65, no. 41, Oct. 2009, pp. 8461-8467. https://doi.org/10.1016/j.tet.2009.08.035.