Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties
Тип публикации: Journal Article
Дата публикации: 1995-03-01
scimago Q2
wos Q1
БС1
SJR: 0.608
CiteScore: 6.7
Impact factor: 3
ISSN: 09680896, 14643391
PubMed ID:
7606391
Organic Chemistry
Drug Discovery
Biochemistry
Molecular Biology
Pharmaceutical Science
Clinical Biochemistry
Molecular Medicine
Краткое описание
Stereochemically defined and epimeric phosphonamidate methyl ester-containing peptide analogues were synthesised and were found to be moderate inhibitors of the HIV-1 proteinase. All of the analogues containing the phosphonamidate ester grouping showed a marked ability to enter cells, as highlighted by the approximate equivalence of the IC50 values for enzyme inhibition in solution and inhibition of HIV-1 replication in virus infected cells.
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ГОСТ
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Camp N. P. et al. Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties // Bioorganic and Medicinal Chemistry. 1995. Vol. 3. No. 3. pp. 297-312.
ГОСТ со всеми авторами (до 50)
Скопировать
Camp N. P., Perrey D. A., Kinchington D., Hawkins P., Gani D. Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties // Bioorganic and Medicinal Chemistry. 1995. Vol. 3. No. 3. pp. 297-312.
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RIS
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TY - JOUR
DO - 10.1016/0968-0896(95)00022-9
UR - https://doi.org/10.1016/0968-0896(95)00022-9
TI - Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties
T2 - Bioorganic and Medicinal Chemistry
AU - Camp, Nicholas P.
AU - Perrey, David A.
AU - Kinchington, Derek
AU - Hawkins, Paul
AU - Gani, David
PY - 1995
DA - 1995/03/01
PB - Elsevier
SP - 297-312
IS - 3
VL - 3
PMID - 7606391
SN - 0968-0896
SN - 1464-3391
ER -
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BibTex (до 50 авторов)
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@article{1995_Camp,
author = {Nicholas P. Camp and David A. Perrey and Derek Kinchington and Paul Hawkins and David Gani},
title = {Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties},
journal = {Bioorganic and Medicinal Chemistry},
year = {1995},
volume = {3},
publisher = {Elsevier},
month = {mar},
url = {https://doi.org/10.1016/0968-0896(95)00022-9},
number = {3},
pages = {297--312},
doi = {10.1016/0968-0896(95)00022-9}
}
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MLA
Скопировать
Camp, Nicholas P., et al. “Synthesis of peptide analogues containing phosphonamidate methyl ester functionality: HIV-1 proteinase inhibitors possessing unique cell uptake properties.” Bioorganic and Medicinal Chemistry, vol. 3, no. 3, Mar. 1995, pp. 297-312. https://doi.org/10.1016/0968-0896(95)00022-9.