Open Access
Open access
volume 13 issue 9 pages 3659-3677

Research advances in peptide‒drug conjugates

Liming Gong 1
Heming Zhao 1
Yanhong Liu 1
Hao Wu 2
Chao Liu 1
Shuangyan Chang 1
Liqing Chen 1
MINGJI JIN 1
Qiming Wang 1
ZHONGGAO GAO 1
Wei Huang 1
Publication typeJournal Article
Publication date2023-09-01
scimago Q1
wos Q1
SJR3.489
CiteScore24.3
Impact factor14.6
ISSN22113835, 22113843
General Pharmacology, Toxicology and Pharmaceutics
Abstract
Peptide‒drug conjugates (PDCs) are drug delivery systems consisting of a drug covalently coupled to a multifunctional peptide via a cleavable linker. As an emerging prodrug strategy, PDCs not only preserve the function and bioactivity of the peptides but also release the drugs responsively with the cleavable property of the linkers. Given the ability to significantly improve the circulation stability and targeting of drugs in vivo and reduce the toxic side effects of drugs, PDCs have already been extensively applied in drug delivery. Herein, we review the types and mechanisms of peptides, linkers and drugs used to construct PDCs, and summarize the clinical applications and challenges of PDC drugs.
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GOST |
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GOST Copy
Gong L. et al. Research advances in peptide‒drug conjugates // Acta Pharmaceutica Sinica B. 2023. Vol. 13. No. 9. pp. 3659-3677.
GOST all authors (up to 50) Copy
Gong L., Zhao H., Liu Y., Wu H., Liu C., Chang S., Chen L., JIN M., Wang Q., GAO Z., Huang W. Research advances in peptide‒drug conjugates // Acta Pharmaceutica Sinica B. 2023. Vol. 13. No. 9. pp. 3659-3677.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1016/j.apsb.2023.02.013
UR - https://doi.org/10.1016/j.apsb.2023.02.013
TI - Research advances in peptide‒drug conjugates
T2 - Acta Pharmaceutica Sinica B
AU - Gong, Liming
AU - Zhao, Heming
AU - Liu, Yanhong
AU - Wu, Hao
AU - Liu, Chao
AU - Chang, Shuangyan
AU - Chen, Liqing
AU - JIN, MINGJI
AU - Wang, Qiming
AU - GAO, ZHONGGAO
AU - Huang, Wei
PY - 2023
DA - 2023/09/01
PB - Elsevier
SP - 3659-3677
IS - 9
VL - 13
PMID - 37719380
SN - 2211-3835
SN - 2211-3843
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2023_Gong,
author = {Liming Gong and Heming Zhao and Yanhong Liu and Hao Wu and Chao Liu and Shuangyan Chang and Liqing Chen and MINGJI JIN and Qiming Wang and ZHONGGAO GAO and Wei Huang},
title = {Research advances in peptide‒drug conjugates},
journal = {Acta Pharmaceutica Sinica B},
year = {2023},
volume = {13},
publisher = {Elsevier},
month = {sep},
url = {https://doi.org/10.1016/j.apsb.2023.02.013},
number = {9},
pages = {3659--3677},
doi = {10.1016/j.apsb.2023.02.013}
}
MLA
Cite this
MLA Copy
Gong, Liming, et al. “Research advances in peptide‒drug conjugates.” Acta Pharmaceutica Sinica B, vol. 13, no. 9, Sep. 2023, pp. 3659-3677. https://doi.org/10.1016/j.apsb.2023.02.013.