3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors
Publication type: Journal Article
Publication date: 2006-01-01
scimago Q2
wos Q2
SJR: 0.472
CiteScore: 5.1
Impact factor: 2.2
ISSN: 0960894X, 14643405
PubMed ID:
16236508
Organic Chemistry
Drug Discovery
Biochemistry
Molecular Biology
Pharmaceutical Science
Clinical Biochemistry
Molecular Medicine
Abstract
The solid-phase supported synthesis and antiphosphatase activity of a series of indolizines are reported. In the course of studies directed toward the discovery of novel scaffolds for medicinal application, we synthesized a series of 3-substituted indolizine-1-carbonitrile derivatives. Some of them displayed activity against MPtpA/MPtpB phosphatases which are involved in infectious diseases. We report here the solid-phase synthesis and antiphosphatase activity of a series of indolizines.
Found
Nothing found, try to update filter.
Found
Nothing found, try to update filter.
Top-30
Journals
|
2
4
6
8
10
12
14
16
|
|
|
Journal of Organic Chemistry
16 publications, 12.7%
|
|
|
Tetrahedron Letters
7 publications, 5.56%
|
|
|
Organic Letters
7 publications, 5.56%
|
|
|
Organic and Biomolecular Chemistry
7 publications, 5.56%
|
|
|
RSC Advances
6 publications, 4.76%
|
|
|
Tetrahedron
5 publications, 3.97%
|
|
|
ChemistrySelect
5 publications, 3.97%
|
|
|
European Journal of Organic Chemistry
5 publications, 3.97%
|
|
|
Advanced Synthesis and Catalysis
3 publications, 2.38%
|
|
|
Journal of Combinatorial Chemistry
3 publications, 2.38%
|
|
|
Chemical Communications
3 publications, 2.38%
|
|
|
Organic Chemistry Frontiers
3 publications, 2.38%
|
|
|
Bioorganic and Medicinal Chemistry Letters
2 publications, 1.59%
|
|
|
Asian Journal of Organic Chemistry
2 publications, 1.59%
|
|
|
Chinese Journal of Chemistry
2 publications, 1.59%
|
|
|
ChemMedChem
2 publications, 1.59%
|
|
|
ACS Combinatorial Science
2 publications, 1.59%
|
|
|
MedChemComm
2 publications, 1.59%
|
|
|
Synthetic Communications
2 publications, 1.59%
|
|
|
Canadian Journal of Chemistry
1 publication, 0.79%
|
|
|
Acta Crystallographica Section E Structure Reports Online
1 publication, 0.79%
|
|
|
Organic Preparations and Procedures International
1 publication, 0.79%
|
|
|
Future Medicinal Chemistry
1 publication, 0.79%
|
|
|
Catalysts
1 publication, 0.79%
|
|
|
Russian Chemical Bulletin
1 publication, 0.79%
|
|
|
Monatshefte fur Chemie
1 publication, 0.79%
|
|
|
Journal of Molecular Structure
1 publication, 0.79%
|
|
|
Medicinal Chemistry Research
1 publication, 0.79%
|
|
|
Pharmacological Reports
1 publication, 0.79%
|
|
|
2
4
6
8
10
12
14
16
|
Publishers
|
5
10
15
20
25
30
|
|
|
American Chemical Society (ACS)
29 publications, 23.02%
|
|
|
Elsevier
27 publications, 21.43%
|
|
|
Royal Society of Chemistry (RSC)
24 publications, 19.05%
|
|
|
Wiley
23 publications, 18.25%
|
|
|
Taylor & Francis
6 publications, 4.76%
|
|
|
Springer Nature
5 publications, 3.97%
|
|
|
Bentham Science Publishers Ltd.
2 publications, 1.59%
|
|
|
Canadian Science Publishing
1 publication, 0.79%
|
|
|
International Union of Crystallography (IUCr)
1 publication, 0.79%
|
|
|
MDPI
1 publication, 0.79%
|
|
|
Pleiades Publishing
1 publication, 0.79%
|
|
|
Oxford University Press
1 publication, 0.79%
|
|
|
The Japan Institute of Heterocyclic Chemistry
1 publication, 0.79%
|
|
|
Walter de Gruyter
1 publication, 0.79%
|
|
|
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 publication, 0.79%
|
|
|
Beilstein-Institut
1 publication, 0.79%
|
|
|
5
10
15
20
25
30
|
- We do not take into account publications without a DOI.
- Statistics recalculated weekly.
Are you a researcher?
Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
126
Total citations:
126
Citations from 2025:
7
(5.56%)
Cite this
GOST |
RIS |
BibTex |
MLA
Cite this
GOST
Copy
Weide T. et al. 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors // Bioorganic and Medicinal Chemistry Letters. 2006. Vol. 16. No. 1. pp. 59-63.
GOST all authors (up to 50)
Copy
Weide T., Arve L., PRINZ H., Waldmann H., Kessler H. 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors // Bioorganic and Medicinal Chemistry Letters. 2006. Vol. 16. No. 1. pp. 59-63.
Cite this
RIS
Copy
TY - JOUR
DO - 10.1016/j.bmcl.2005.09.051
UR - https://doi.org/10.1016/j.bmcl.2005.09.051
TI - 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors
T2 - Bioorganic and Medicinal Chemistry Letters
AU - Weide, Timo
AU - Arve, Lars
AU - PRINZ, Heino
AU - Waldmann, Herbert
AU - Kessler, H.
PY - 2006
DA - 2006/01/01
PB - Elsevier
SP - 59-63
IS - 1
VL - 16
PMID - 16236508
SN - 0960-894X
SN - 1464-3405
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2006_Weide,
author = {Timo Weide and Lars Arve and Heino PRINZ and Herbert Waldmann and H. Kessler},
title = {3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors},
journal = {Bioorganic and Medicinal Chemistry Letters},
year = {2006},
volume = {16},
publisher = {Elsevier},
month = {jan},
url = {https://doi.org/10.1016/j.bmcl.2005.09.051},
number = {1},
pages = {59--63},
doi = {10.1016/j.bmcl.2005.09.051}
}
Cite this
MLA
Copy
Weide, Timo, et al. “3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors.” Bioorganic and Medicinal Chemistry Letters, vol. 16, no. 1, Jan. 2006, pp. 59-63. https://doi.org/10.1016/j.bmcl.2005.09.051.