Bioorganic and Medicinal Chemistry Letters

, том 16 , издание 1 , страницы 59-63

3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors

Timo Weide ¹

Lars Arve ²

Heino PRINZ ³

Herbert Waldmann ³

H. Kessler ¹

Скрыть аффилиации авторов Показать аффилиации авторов: 3 аффилиации

Department Chemie, Lehrstuhl II für Organische Chemie, Technische Universität München, Lichtenbergstr. 4, D-85747 Garching, Germany. |

Max Planck Institute of Molecular Physiology, Max Planck Society |

Abt. IV: Chemische Biologie, Max Planck Institute of Molecular Physiology, Max Planck Society |

Тип публикации: Journal Article

Дата публикации: 2006-01-01

Elsevier

Bioorganic and Medicinal Chemistry Letters

scimago Q2

wos Q2

БС2

SJR: 0.472

CiteScore: 5.1

Impact factor: 2.2

ISSN: 0960894X, 14643405

DOI: 10.1016/j.bmcl.2005.09.051

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PubMed ID: 16236508

Organic Chemistry

Drug Discovery

Biochemistry

Molecular Biology

Pharmaceutical Science

Clinical Biochemistry

Molecular Medicine

Краткое описание

The solid-phase supported synthesis and antiphosphatase activity of a series of indolizines are reported. In the course of studies directed toward the discovery of novel scaffolds for medicinal application, we synthesized a series of 3-substituted indolizine-1-carbonitrile derivatives. Some of them displayed activity against MPtpA/MPtpB phosphatases which are involved in infectious diseases. We report here the solid-phase synthesis and antiphosphatase activity of a series of indolizines.

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Weide T. et al. 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors // Bioorganic and Medicinal Chemistry Letters. 2006. Vol. 16. No. 1. pp. 59-63.

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Weide T., Arve L., PRINZ H., Waldmann H., Kessler H. 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors // Bioorganic and Medicinal Chemistry Letters. 2006. Vol. 16. No. 1. pp. 59-63.

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RIS Скопировать

TY - JOUR

DO - 10.1016/j.bmcl.2005.09.051

UR - https://doi.org/10.1016/j.bmcl.2005.09.051

TI - 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors

T2 - Bioorganic and Medicinal Chemistry Letters

AU - Weide, Timo

AU - Arve, Lars

AU - PRINZ, Heino

AU - Waldmann, Herbert

AU - Kessler, H.

PY - 2006

DA - 2006/01/01

PB - Elsevier

SP - 59-63

IS - 1

VL - 16

PMID - 16236508

SN - 0960-894X

SN - 1464-3405

ER -

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@article{2006_Weide,

author = {Timo Weide and Lars Arve and Heino PRINZ and Herbert Waldmann and H. Kessler},

title = {3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors},

journal = {Bioorganic and Medicinal Chemistry Letters},

year = {2006},

volume = {16},

publisher = {Elsevier},

month = {jan},

url = {https://doi.org/10.1016/j.bmcl.2005.09.051},

number = {1},

pages = {59--63},

doi = {10.1016/j.bmcl.2005.09.051}

}

MLA

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MLA Скопировать

Weide, Timo, et al. “3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors.” Bioorganic and Medicinal Chemistry Letters, vol. 16, no. 1, Jan. 2006, pp. 59-63. https://doi.org/10.1016/j.bmcl.2005.09.051.

Издатель

Elsevier

Журнал

Bioorganic and Medicinal Chemistry Letters

scimago Q2

wos Q2

БС2

SJR

0.472

CiteScore

5.1

Impact factor

2.2

ISSN

0960894X (Print)

14643405 (Electronic)