Bioorganic and Medicinal Chemistry Letters, volume 26, issue 10, pages 2455-2458
A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity
E.V. Shchegol’kov
1
,
Irina V Shchur
1
,
Yanina V. Burgart
1
,
Victor Saloutin
1
,
Sergey Yu Solodnikov
2
,
Olga P Krasnykh
2
,
Marionella A. Kravchenko
3
Publication type: Journal Article
Publication date: 2016-05-01
Quartile SCImago
Q2
Quartile WOS
Q2
Impact factor: 2.7
ISSN: 0960894X, 14643405
Organic Chemistry
Drug Discovery
Biochemistry
Molecular Biology
Pharmaceutical Science
Clinical Biochemistry
Molecular Medicine
Abstract
We have developed the practical method for polyfluorosalicylic acids synthesis via nucleophilic ortho-mono-substitution of fluorine atom with magnesium methoxide. We have managed to increase the yield of targeted polyfluorosalicylic acids from good to quantitative. We have studied the tuberculostatic activity of polyfluorosalicylic acids. It has been found that minimum inhibitory concentration (MIC) of compounds is from 0.7 to 6.5μg/mL depending on the structure.
Top-30
Citations by journals
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1
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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1 publication, 11.11%
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Russian Chemical Reviews
1 publication, 11.11%
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1
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Citations by publishers
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1
2
3
4
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Elsevier
4 publications, 44.44%
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Wiley
2 publications, 22.22%
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Multidisciplinary Digital Publishing Institute (MDPI)
1 publication, 11.11%
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American Institute of Physics (AIP)
1 publication, 11.11%
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Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii
1 publication, 11.11%
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- We do not take into account publications without a DOI.
- Statistics recalculated only for publications connected to researchers, organizations and labs registered on the platform.
- Statistics recalculated weekly.
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Shchegol’kov E. et al. A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity // Bioorganic and Medicinal Chemistry Letters. 2016. Vol. 26. No. 10. pp. 2455-2458.
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Shchegol’kov E., Shchur I. V., Burgart Y. V., Saloutin V., Solodnikov S. Yu., Krasnykh O. P., Kravchenko M. A. A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity // Bioorganic and Medicinal Chemistry Letters. 2016. Vol. 26. No. 10. pp. 2455-2458.
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TY - JOUR
DO - 10.1016/j.bmcl.2016.03.107
UR - https://doi.org/10.1016/j.bmcl.2016.03.107
TI - A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity
T2 - Bioorganic and Medicinal Chemistry Letters
AU - Shchegol’kov, E.V.
AU - Shchur, Irina V
AU - Burgart, Yanina V.
AU - Saloutin, Victor
AU - Solodnikov, Sergey Yu
AU - Krasnykh, Olga P
AU - Kravchenko, Marionella A.
PY - 2016
DA - 2016/05/01 00:00:00
PB - Elsevier
SP - 2455-2458
IS - 10
VL - 26
SN - 0960-894X
SN - 1464-3405
ER -
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@article{2016_Shchegol’kov,
author = {E.V. Shchegol’kov and Irina V Shchur and Yanina V. Burgart and Victor Saloutin and Sergey Yu Solodnikov and Olga P Krasnykh and Marionella A. Kravchenko},
title = {A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity},
journal = {Bioorganic and Medicinal Chemistry Letters},
year = {2016},
volume = {26},
publisher = {Elsevier},
month = {may},
url = {https://doi.org/10.1016/j.bmcl.2016.03.107},
number = {10},
pages = {2455--2458},
doi = {10.1016/j.bmcl.2016.03.107}
}
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Shchegol’kov, E.V., et al. “A convenient and efficient approach to polyfluorosalicylic acids and their tuberculostatic activity.” Bioorganic and Medicinal Chemistry Letters, vol. 26, no. 10, May. 2016, pp. 2455-2458. https://doi.org/10.1016/j.bmcl.2016.03.107.
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