Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives
Feng Yun Li
1
,
Xiaofeng Guo
1
,
Zhijin Fan
1
,
Yuan Zhang
1
,
Guang Ning Zong
1
,
Xiaolin Qian
1
,
Liu Yong Ma
1
,
Lei Chen
1
,
Yujie Zhu
1
,
Tatiana Kalinina
2
,
Yury Yu. Morzherin
2
,
1
Тип публикации: Journal Article
Дата публикации: 2015-10-01
scimago Q1
wos Q1
БС1
SJR: 1.677
CiteScore: 15.7
Impact factor: 8.9
ISSN: 10018417, 18785964
General Chemistry
Краткое описание
A series of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives were designed and synthesized. Their structures were confirmed by melting points, IR, 1H NMR, 13C NMR, and HRMS or elemental analysis. Biological activities of all title compounds including fungicidal activity and antivirus activity were evaluated systematically. Preliminary bioassays indicated that these compounds exhibited good fungicidal activity at 50 μg/mL, compounds 4b and 4i exhibited over 50% activity against six fungi tested. Most compounds showed good activity against TMV with different models in vivo at 100 μg/mL. Compounds 4c and 4e stood out with high effects against TMV in vivo in all models tested, including protective, inactivative, curative, and inductive activities. These data demonstrate a new strategy for fungi and virus control.
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Li F. Y. et al. Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives // Chinese Chemical Letters. 2015. Vol. 26. No. 10. pp. 1315-1318.
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Li F. Y., Guo X., Fan Z., Zhang Y., Zong G. N., Qian X., Ma L. Y., Chen L., Zhu Y., Kalinina T., Morzherin Y. Y., Belskaya N. P. Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives // Chinese Chemical Letters. 2015. Vol. 26. No. 10. pp. 1315-1318.
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TY - JOUR
DO - 10.1016/j.cclet.2015.05.040
UR - https://doi.org/10.1016/j.cclet.2015.05.040
TI - Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives
T2 - Chinese Chemical Letters
AU - Li, Feng Yun
AU - Guo, Xiaofeng
AU - Fan, Zhijin
AU - Zhang, Yuan
AU - Zong, Guang Ning
AU - Qian, Xiaolin
AU - Ma, Liu Yong
AU - Chen, Lei
AU - Zhu, Yujie
AU - Kalinina, Tatiana
AU - Morzherin, Yury Yu.
AU - Belskaya, Nataliya P.
PY - 2015
DA - 2015/10/01
PB - Elsevier
SP - 1315-1318
IS - 10
VL - 26
SN - 1001-8417
SN - 1878-5964
ER -
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@article{2015_Li,
author = {Feng Yun Li and Xiaofeng Guo and Zhijin Fan and Yuan Zhang and Guang Ning Zong and Xiaolin Qian and Liu Yong Ma and Lei Chen and Yujie Zhu and Tatiana Kalinina and Yury Yu. Morzherin and Nataliya P. Belskaya},
title = {Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives},
journal = {Chinese Chemical Letters},
year = {2015},
volume = {26},
publisher = {Elsevier},
month = {oct},
url = {https://doi.org/10.1016/j.cclet.2015.05.040},
number = {10},
pages = {1315--1318},
doi = {10.1016/j.cclet.2015.05.040}
}
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MLA
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Li, Feng Yun, et al. “Synthesis and biological activities of novel 2-amino-1,3-thiazole-4-carboxylic acid derivatives.” Chinese Chemical Letters, vol. 26, no. 10, Oct. 2015, pp. 1315-1318. https://doi.org/10.1016/j.cclet.2015.05.040.