Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides
Тип публикации: Journal Article
Дата публикации: 2009-08-01
scimago Q1
wos Q1
БС1
SJR: 1.151
CiteScore: 11.7
Impact factor: 5.9
ISSN: 02235234, 17683254
PubMed ID:
19371979
Organic Chemistry
Drug Discovery
General Medicine
Pharmacology
Краткое описание
A series of 4-substituted imidazolyl-2,6-dimethyl-N(3),N(5)-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides were prepared. They were screened as antitubercular agents against Mycobacterium tuberculosis H(37)Rv. Minimum inhibitory concentrations (MICs) were determined using agar proportion method. Compound 3i with 1-benzyl-2-methylthio-1H-imidazole-5-yl substituent at C-4 position and 4'-chloromophenyl group at C-3 and C-5 positions of the 1,4-dihydropyridine ring was the most potent one among the tested compounds. It was as potent as rifampicin against M. tuberculosis H(37)RV. Compound 3l also was an active antitubercular agent with the same substituent as compound 3i at the C-4 position and 3'-pyridyl group at C-3 and C-5 positions of the 1,4-dihydropyridine ring.
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Fassihi A. et al. Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides // European Journal of Medicinal Chemistry. 2009. Vol. 44. No. 8. pp. 3253-3258.
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Fassihi A., Azadpour Z., Delbari N., Saghaie L., Memarian H. R., Sabet R., Alborzi A., Miri R., Pourabbas B., Mardaneh J. Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides // European Journal of Medicinal Chemistry. 2009. Vol. 44. No. 8. pp. 3253-3258.
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TY - JOUR
DO - 10.1016/j.ejmech.2009.03.027
UR - https://doi.org/10.1016/j.ejmech.2009.03.027
TI - Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides
T2 - European Journal of Medicinal Chemistry
AU - Fassihi, Afshin
AU - Azadpour, Zahra
AU - Delbari, Neda
AU - Saghaie, Lotfollah
AU - Memarian, Hamid R
AU - Sabet, Razieh
AU - Alborzi, Abdolvahab
AU - Miri, Ramin
AU - Pourabbas, Bahman
AU - Mardaneh, Jalal
PY - 2009
DA - 2009/08/01
PB - Elsevier
SP - 3253-3258
IS - 8
VL - 44
PMID - 19371979
SN - 0223-5234
SN - 1768-3254
ER -
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@article{2009_Fassihi,
author = {Afshin Fassihi and Zahra Azadpour and Neda Delbari and Lotfollah Saghaie and Hamid R Memarian and Razieh Sabet and Abdolvahab Alborzi and Ramin Miri and Bahman Pourabbas and Jalal Mardaneh},
title = {Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides},
journal = {European Journal of Medicinal Chemistry},
year = {2009},
volume = {44},
publisher = {Elsevier},
month = {aug},
url = {https://doi.org/10.1016/j.ejmech.2009.03.027},
number = {8},
pages = {3253--3258},
doi = {10.1016/j.ejmech.2009.03.027}
}
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MLA
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Fassihi, Afshin, et al. “Synthesis and antitubercular activity of novel 4-substituted imidazolyl-2,6-dimethyl-N3,N5-bisaryl-1,4-dihydropyridine-3,5-dicarboxamides.” European Journal of Medicinal Chemistry, vol. 44, no. 8, Aug. 2009, pp. 3253-3258. https://doi.org/10.1016/j.ejmech.2009.03.027.