Open Access
Cocrystal screening of hydroxybenzamides with benzoic acid derivatives: A comparative study of thermal and solution-based methods
Тип публикации: Journal Article
Дата публикации: 2014-12-01
scimago Q1
wos Q1
БС1
SJR: 0.827
CiteScore: 9.1
Impact factor: 4.7
ISSN: 09280987, 18790720
PubMed ID:
25218047
Pharmaceutical Science
Краткое описание
The main problem occurring at the early stages of cocrystal search is the choice of an effective screening technique. Among the most popular techniques of obtaining cocrystals are crystallization from solution, crystallization from melt and solvent-drop grinding. This paper represents a comparative analysis of the following screening techniques: DSC cocrystal screening method, thermal microscopy and saturation temperature method. The efficiency of different techniques of cocrystal screening was checked in 18 systems. Benzamide and benzoic acid derivatives were chosen as model systems due to their ability to form acid-amide supramolecular heterosynthon. The screening has confirmed the formation of 6 new cocrystals. The screening by the saturation temperature method has the highest screen-out rate but the smallest range of application. DSC screening has a satisfactory accuracy and allows screening over a short time. Thermal microscopy is most efficient as an additional technique used to interpret ambiguous DSC screening results. The study also included an analysis of the influence of solvent type and component solubility on cocrystal formation.
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Manin A. N. et al. Cocrystal screening of hydroxybenzamides with benzoic acid derivatives: A comparative study of thermal and solution-based methods // European Journal of Pharmaceutical Sciences. 2014. Vol. 65. pp. 56-64.
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Manin A. N., Voronin A., Drozd K. V., Manin N. G., Bauer-Brandl A., Perlovich G. Cocrystal screening of hydroxybenzamides with benzoic acid derivatives: A comparative study of thermal and solution-based methods // European Journal of Pharmaceutical Sciences. 2014. Vol. 65. pp. 56-64.
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TY - JOUR
DO - 10.1016/j.ejps.2014.09.003
UR - https://doi.org/10.1016/j.ejps.2014.09.003
TI - Cocrystal screening of hydroxybenzamides with benzoic acid derivatives: A comparative study of thermal and solution-based methods
T2 - European Journal of Pharmaceutical Sciences
AU - Manin, Alex N
AU - Voronin, Alexander
AU - Drozd, Ksenia V.
AU - Manin, Nikolay G
AU - Bauer-Brandl, Annette
AU - Perlovich, German
PY - 2014
DA - 2014/12/01
PB - Elsevier
SP - 56-64
VL - 65
PMID - 25218047
SN - 0928-0987
SN - 1879-0720
ER -
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@article{2014_Manin,
author = {Alex N Manin and Alexander Voronin and Ksenia V. Drozd and Nikolay G Manin and Annette Bauer-Brandl and German Perlovich},
title = {Cocrystal screening of hydroxybenzamides with benzoic acid derivatives: A comparative study of thermal and solution-based methods},
journal = {European Journal of Pharmaceutical Sciences},
year = {2014},
volume = {65},
publisher = {Elsevier},
month = {dec},
url = {https://doi.org/10.1016/j.ejps.2014.09.003},
pages = {56--64},
doi = {10.1016/j.ejps.2014.09.003}
}