Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives
Publication type: Journal Article
Publication date: 2004-09-01
scimago Q3
wos Q3
SJR: 0.333
CiteScore: 3.7
Impact factor: 1.9
ISSN: 00221139, 18733328
Organic Chemistry
Biochemistry
Inorganic Chemistry
Physical and Theoretical Chemistry
Environmental Chemistry
Abstract
Nine novel 2-methyl-4-trifluoromethylthiazole-5-carboxamide derivatives were designed and synthesized utilizing ethyl 4,4,4-trifluoroacetoacetate as a starting material. Subsequently, the biological activity of the compounds was evaluated in the greenhouse. Results indicated that all of the compounds have some fungicidal and insecticidal activity but no herbicidal activity. Compound 1 has fungicidal activity with 90% control of tomato late blight at 375 g ai/ha, while two compounds 2F and 2H show insecticidal activity with 80 and 100% control, respectively, against potato leafhopper at 600 g ai/ha.
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Total citations:
41
Citations from 2025:
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(2.44%)
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GOST
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Liu C., Li Z., Zhong B. Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives // Journal of Fluorine Chemistry. 2004. Vol. 125. No. 9. pp. 1287-1290.
GOST all authors (up to 50)
Copy
Liu C., Li Z., Zhong B. Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives // Journal of Fluorine Chemistry. 2004. Vol. 125. No. 9. pp. 1287-1290.
Cite this
RIS
Copy
TY - JOUR
DO - 10.1016/j.jfluchem.2004.03.006
UR - https://doi.org/10.1016/j.jfluchem.2004.03.006
TI - Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives
T2 - Journal of Fluorine Chemistry
AU - Liu, Changling
AU - Li, Zheng-Ming
AU - Zhong, Bin
PY - 2004
DA - 2004/09/01
PB - Elsevier
SP - 1287-1290
IS - 9
VL - 125
SN - 0022-1139
SN - 1873-3328
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2004_Liu,
author = {Changling Liu and Zheng-Ming Li and Bin Zhong},
title = {Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives},
journal = {Journal of Fluorine Chemistry},
year = {2004},
volume = {125},
publisher = {Elsevier},
month = {sep},
url = {https://doi.org/10.1016/j.jfluchem.2004.03.006},
number = {9},
pages = {1287--1290},
doi = {10.1016/j.jfluchem.2004.03.006}
}
Cite this
MLA
Copy
Liu, Changling, et al. “Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives.” Journal of Fluorine Chemistry, vol. 125, no. 9, Sep. 2004, pp. 1287-1290. https://doi.org/10.1016/j.jfluchem.2004.03.006.