Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling
Тип публикации: Journal Article
Дата публикации: 2010-09-01
scimago Q3
wos Q3
БС1
SJR: 0.305
CiteScore: 3
Impact factor: 1.7
ISSN: 09599436, 1364551X
General Chemistry
Краткое описание
A set of novel fragment-like catechol derivatives were identified as EphA2 inhibitors and were further profiled against a panel of 19 tyrosine kinases. In addition to EphA2, the recovered hits were active against EGFR, FGFR1, FGFR2, Abl and PDGFR-a, and according to molecular modelling studies catechol moiety was capable of forming two or more correlated hydrogen bonds with the kinase hinge region, suggesting prospects of its further optimization as an EphA2 inhibitor.
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Stroylov V. et al. Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling // Mendeleev Communications. 2010. Vol. 20. No. 5. pp. 263-265.
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Stroylov V., Rakitina T. V., Novikov F., Stroganov O. V., Chilova G. G., Lipkin A. V. Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling // Mendeleev Communications. 2010. Vol. 20. No. 5. pp. 263-265.
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TY - JOUR
DO - 10.1016/j.mencom.2010.09.007
UR - https://doi.org/10.1016/j.mencom.2010.09.007
TI - Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling
T2 - Mendeleev Communications
AU - Stroylov, Victor
AU - Rakitina, Tatiana V.
AU - Novikov, Fedor
AU - Stroganov, Oleg V.
AU - Chilova, Ghermes G
AU - Lipkin, Aleksey V.
PY - 2010
DA - 2010/09/01
PB - OOO Zhurnal "Mendeleevskie Soobshcheniya"
SP - 263-265
IS - 5
VL - 20
SN - 0959-9436
SN - 1364-551X
ER -
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@article{2010_Stroylov,
author = {Victor Stroylov and Tatiana V. Rakitina and Fedor Novikov and Oleg V. Stroganov and Ghermes G Chilova and Aleksey V. Lipkin},
title = {Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling},
journal = {Mendeleev Communications},
year = {2010},
volume = {20},
publisher = {OOO Zhurnal "Mendeleevskie Soobshcheniya"},
month = {sep},
url = {https://doi.org/10.1016/j.mencom.2010.09.007},
number = {5},
pages = {263--265},
doi = {10.1016/j.mencom.2010.09.007}
}
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MLA
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Stroylov, Victor, et al. “Novel fragment-like inhibitors of EphA2 obtained by experimental screening and modelling.” Mendeleev Communications, vol. 20, no. 5, Sep. 2010, pp. 263-265. https://doi.org/10.1016/j.mencom.2010.09.007.