Mendeleev Communications

, volume 28 , issue 4 , pages 393-395

New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents

Egor V. Verbitskiy ^{1, 2}

Svetlana A Baskakova ³

Natalya A Gerasimova ⁴

Natalya P Evstigneeva ⁴

Natalya V Zilberberg ⁴

Nikolay V Kungurov ⁴

Marionella A. Kravchenko ⁵

Gennady L. Rusinov ^{1, 2}

Oleg N Chupakhina ¹

Valery Charushin ^{1, 2}

Hide authors affiliations Show authors affiliations: 5 affiliations

Institute of Chemical Engineering, Ural Federal University, 620002 Ekaterinburg, Russian Federation |

I. Ya. Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 620990 Ekaterinburg, Russian Federation |

I. Ya. Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 620990, Ekaterinburg, Russian Federation |

⁴

Ural Research Institute for Dermatology, Venereology and Immunopathology, 620076 Ekaterinburg, Russian Federation |

⁵

Ural Research Institute for Phthisiopulmonology, 620039 Ekaterinburg, Russian Federation |

Publication type: Journal Article

Publication date: 2018-07-01

OOO Zhurnal "Mendeleevskie Soobshcheniya"

Mendeleev Communications

scimago Q3

wos Q3

SJR: 0.305

CiteScore: 3.0

Impact factor: 1.7

ISSN: 09599436, 1364551X

DOI: 10.1016/j.mencom.2018.07.017

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General Chemistry

Abstract

A facile synthetic approach to 5-arylamino-4-(5-nitrofuran- 2-yl)pyrimidines by the Buchwald–Hartwig cross-coupling with various anilines has been developed. All synthesized compounds demonstrated a significant level of in vitro antibacterial activity against Neisseria gonorrhoeae, Streptococcus pyogene and Staphylococcus aureus, including their drug-resistant strains, which is much higher than that of the commercial drug Spectinomycin.

Found

1 citation

Osolodkin Dmitry

🥼 🤝

PhD in Chemistry

80 publications, 1 728 citations

h-index: 23

Sechenov First Moscow State Medical University

M.P. Chumakov Federal Scientific Center for Research and Development of Immunobiological Drugs of the Russian Academy of Sciences

1 citation

Varaksin Mikhail

DSc in Chemistry

79 publications, 829 citations, 12 reviews

h-index: 18

Postovsky Institute of Organic Synthesis of the Ural Branch of the Russian Academy of Sciences

Ural Federal University

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Verbitskiy E. V. et al. New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents // Mendeleev Communications. 2018. Vol. 28. No. 4. pp. 393-395.

GOST all authors (up to 50) Copy

Verbitskiy E. V., Baskakova S. A., Gerasimova N. A., Evstigneeva N. P., Zilberberg N. V., Kungurov N. V., Kravchenko M. A., Rusinov G. L., Chupakhina O. N., Charushin V. New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents // Mendeleev Communications. 2018. Vol. 28. No. 4. pp. 393-395.

RIS |

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RIS Copy

TY - JOUR

DO - 10.1016/j.mencom.2018.07.017

UR - https://doi.org/10.1016/j.mencom.2018.07.017

TI - New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents

T2 - Mendeleev Communications

AU - Verbitskiy, Egor V.

AU - Baskakova, Svetlana A

AU - Gerasimova, Natalya A

AU - Evstigneeva, Natalya P

AU - Zilberberg, Natalya V

AU - Kungurov, Nikolay V

AU - Kravchenko, Marionella A.

AU - Rusinov, Gennady L.

AU - Chupakhina, Oleg N

AU - Charushin, Valery

PY - 2018

DA - 2018/07/01

PB - OOO Zhurnal "Mendeleevskie Soobshcheniya"

SP - 393-395

IS - 4

VL - 28

SN - 0959-9436

SN - 1364-551X

ER -

BibTex |

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BibTex (up to 50 authors) Copy

@article{2018_Verbitskiy,

author = {Egor V. Verbitskiy and Svetlana A Baskakova and Natalya A Gerasimova and Natalya P Evstigneeva and Natalya V Zilberberg and Nikolay V Kungurov and Marionella A. Kravchenko and Gennady L. Rusinov and Oleg N Chupakhina and Valery Charushin},

title = {New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents},

journal = {Mendeleev Communications},

year = {2018},

volume = {28},

publisher = {OOO Zhurnal "Mendeleevskie Soobshcheniya"},

month = {jul},

url = {https://doi.org/10.1016/j.mencom.2018.07.017},

number = {4},

pages = {393--395},

doi = {10.1016/j.mencom.2018.07.017}

}

MLA

Cite this

MLA Copy

Verbitskiy, Egor V., et al. “New 5-arylamino-4-(5-nitrofuran-2-yl)pyrimidines as promising antibacterial agents.” Mendeleev Communications, vol. 28, no. 4, Jul. 2018, pp. 393-395. https://doi.org/10.1016/j.mencom.2018.07.017.

Publisher

OOO Zhurnal "Mendeleevskie Soobshcheniya"

Journal

Mendeleev Communications

scimago Q3

wos Q3

SJR

0.305

CiteScore

3.0

Impact factor

1.7

ISSN

09599436 (Print)

1364551X (Electronic)