A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores
Publication type: Journal Article
Publication date: 2019-03-01
scimago Q3
wos Q3
SJR: 0.305
CiteScore: 3.0
Impact factor: 1.7
ISSN: 09599436, 1364551X
General Chemistry
Abstract
A series of combretastatin analogues, diarylpyrazoles and diarylisoxazoles, have been synthesized and evaluated for their antimitotic tubulin-binding activity using the phenotypic sea urchin (Paracentrotus lividus) embryo assay. One pyrazole analogue and four isoxazole analogues have been identified as potent antimitotic agents comparable with combretastatins A-2 and A-4, with the lowest observable effective concentration of 1–10 nmol dm−3 for cleavage alteration of the test embryos.
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Tsyganov D. V. et al. A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores // Mendeleev Communications. 2019. Vol. 29. No. 2. pp. 163-165.
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Tsyganov D. V., Semenova M., Konyushkin L. D., Ushkarov V. I., Raihstat M. M., Semenov V. A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores // Mendeleev Communications. 2019. Vol. 29. No. 2. pp. 163-165.
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TY - JOUR
DO - 10.1016/j.mencom.2019.03.015
UR - https://doi.org/10.1016/j.mencom.2019.03.015
TI - A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores
T2 - Mendeleev Communications
AU - Tsyganov, Dmitry V
AU - Semenova, Marina
AU - Konyushkin, Leonid D
AU - Ushkarov, Vladimir I
AU - Raihstat, Mikhail M
AU - Semenov, Victor
PY - 2019
DA - 2019/03/01
PB - OOO Zhurnal "Mendeleevskie Soobshcheniya"
SP - 163-165
IS - 2
VL - 29
SN - 0959-9436
SN - 1364-551X
ER -
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BibTex (up to 50 authors)
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@article{2019_Tsyganov,
author = {Dmitry V Tsyganov and Marina Semenova and Leonid D Konyushkin and Vladimir I Ushkarov and Mikhail M Raihstat and Victor Semenov},
title = {A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores},
journal = {Mendeleev Communications},
year = {2019},
volume = {29},
publisher = {OOO Zhurnal "Mendeleevskie Soobshcheniya"},
month = {mar},
url = {https://doi.org/10.1016/j.mencom.2019.03.015},
number = {2},
pages = {163--165},
doi = {10.1016/j.mencom.2019.03.015}
}
Cite this
MLA
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Tsyganov, Dmitry V., et al. “A convenient synthesis of cis-restricted combretastatin analogues with pyrazole and isoxazole cores.” Mendeleev Communications, vol. 29, no. 2, Mar. 2019, pp. 163-165. https://doi.org/10.1016/j.mencom.2019.03.015.