Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity
Egor V. Verbitskiy
1, 2
,
Svetlana A Baskakova
2
,
Danila V Belyaev
2
,
Diana V. Vakhrusheva
3
,
Natalya I. Eremeeva
3
,
Gennady L. Rusinov
1, 2
,
Valery Charushin
1, 2
1
Publication type: Journal Article
Publication date: 2021-03-31
scimago Q3
wos Q3
SJR: 0.305
CiteScore: 3.0
Impact factor: 1.7
ISSN: 09599436, 1364551X
General Chemistry
Abstract
The Buchwald–Hartwig cross-coupling of 5-bromo-4-(furan-2-yl)pyrimidine with various anilines afforded the corresponding new 5-(arylamino)pyrimidines, the reaction being accelerated by microwave irradiation. Most of the obtained compounds proved to possess a high bacteriostatic in vitro effect against Mycobacterium tuberculosis H37Rv, Neisseria gonorrhoeae, and Staphylococcus aureus including Methicillin-resistant strain, which is stronger than that of the commercial drug Spectinomycin.
Found
Nothing found, try to update filter.
Found
Nothing found, try to update filter.
Top-30
Journals
|
1
2
3
4
|
|
|
Mendeleev Communications
4 publications, 30.77%
|
|
|
ChemistrySelect
1 publication, 7.69%
|
|
|
Biomedicines
1 publication, 7.69%
|
|
|
MolBank
1 publication, 7.69%
|
|
|
Biomolecules
1 publication, 7.69%
|
|
|
Progress in Heterocyclic Chemistry
1 publication, 7.69%
|
|
|
Current Organic Synthesis
1 publication, 7.69%
|
|
|
International Journal of Molecular Sciences
1 publication, 7.69%
|
|
|
Advances in Heterocyclic Chemistry
1 publication, 7.69%
|
|
|
Russian Chemical Bulletin
1 publication, 7.69%
|
|
|
1
2
3
4
|
Publishers
|
1
2
3
4
|
|
|
MDPI
4 publications, 30.77%
|
|
|
OOO Zhurnal "Mendeleevskie Soobshcheniya"
4 publications, 30.77%
|
|
|
Elsevier
2 publications, 15.38%
|
|
|
Wiley
1 publication, 7.69%
|
|
|
Bentham Science Publishers Ltd.
1 publication, 7.69%
|
|
|
Springer Nature
1 publication, 7.69%
|
|
|
1
2
3
4
|
- We do not take into account publications without a DOI.
- Statistics recalculated weekly.
Are you a researcher?
Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
13
Total citations:
13
Citations from 2025:
1
(7.69%)
Cite this
GOST |
RIS |
BibTex |
MLA
Cite this
GOST
Copy
Verbitskiy E. V. et al. Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity // Mendeleev Communications. 2021. Vol. 31. No. 2. pp. 210-212.
GOST all authors (up to 50)
Copy
Verbitskiy E. V., Baskakova S. A., Belyaev D. V., Vakhrusheva D. V., Eremeeva N. I., Rusinov G. L., Charushin V. Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity // Mendeleev Communications. 2021. Vol. 31. No. 2. pp. 210-212.
Cite this
RIS
Copy
TY - JOUR
DO - 10.1016/j.mencom.2021.03.021
UR - https://doi.org/10.1016/j.mencom.2021.03.021
TI - Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity
T2 - Mendeleev Communications
AU - Verbitskiy, Egor V.
AU - Baskakova, Svetlana A
AU - Belyaev, Danila V
AU - Vakhrusheva, Diana V.
AU - Eremeeva, Natalya I.
AU - Rusinov, Gennady L.
AU - Charushin, Valery
PY - 2021
DA - 2021/03/31
PB - OOO Zhurnal "Mendeleevskie Soobshcheniya"
SP - 210-212
IS - 2
VL - 31
SN - 0959-9436
SN - 1364-551X
ER -
Cite this
BibTex (up to 50 authors)
Copy
@article{2021_Verbitskiy,
author = {Egor V. Verbitskiy and Svetlana A Baskakova and Danila V Belyaev and Diana V. Vakhrusheva and Natalya I. Eremeeva and Gennady L. Rusinov and Valery Charushin},
title = {Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity},
journal = {Mendeleev Communications},
year = {2021},
volume = {31},
publisher = {OOO Zhurnal "Mendeleevskie Soobshcheniya"},
month = {mar},
url = {https://doi.org/10.1016/j.mencom.2021.03.021},
number = {2},
pages = {210--212},
doi = {10.1016/j.mencom.2021.03.021}
}
Cite this
MLA
Copy
Verbitskiy, Egor V., et al. “Renaissance of 4-(5-nitrofuran-2-yl)-5-arylamino substituted pyrimidines: microwave-assisted synthesis and antitubercular activity.” Mendeleev Communications, vol. 31, no. 2, Mar. 2021, pp. 210-212. https://doi.org/10.1016/j.mencom.2021.03.021.