том 33 издание 4 страницы 448-450

An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold

Тип публикацииJournal Article
Дата публикации2023-07-17
scimago Q3
wos Q3
БС1
SJR0.305
CiteScore3.0
Impact factor1.7
ISSN09599436, 1364551X
General Chemistry
Краткое описание
Spirocyclization of morpholinium 3-[(aryl)(1,3-dimethyl-2,4,6-trioxohexahydropyrimidin-5-yl)methyl]-6-methyl-2-oxo-2H-pyran-4-olate by the action of sodium acetate-N-bromosuccinimide system in ethanol at room temperature results in spiro[furo[3,2-c]pyran-2,5’-pyrimidine] derivatives in 92–98% yields, the protocol allowing to avoid column chromatography purification. This new highly efficient and facile procedure is a convenient way to substituted unsymmetrical spiro scaffold containing pyrimidine-2,4,6-trione and 2,3-dihydro-4H-furo[3,2-c]pyran-4-one fragments promising for biomedical applications.
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Russian Chemical Bulletin
1 публикация, 25%
Journal of Heterocyclic Chemistry
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MolBank
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Mendeleev Communications
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Springer Nature
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OOO Zhurnal "Mendeleevskie Soobshcheniya"
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ГОСТ |
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Elinson M. N. et al. An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold // Mendeleev Communications. 2023. Vol. 33. No. 4. pp. 448-450.
ГОСТ со всеми авторами (до 50) Скопировать
Elinson M. N., Vereshchagin A. N., Ryzhkova Y. E., Karpenko K. A., Kalashnikova V. M., Egorov M. P. An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold // Mendeleev Communications. 2023. Vol. 33. No. 4. pp. 448-450.
RIS |
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TY - JOUR
DO - 10.1016/j.mencom.2023.06.002
UR - https://doi.org/10.1016/j.mencom.2023.06.002
TI - An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold
T2 - Mendeleev Communications
AU - Elinson, M. N.
AU - Vereshchagin, Anatoly N.
AU - Ryzhkova, Yuliya E.
AU - Karpenko, Kirill A
AU - Kalashnikova, Varvara M
AU - Egorov, M. P.
PY - 2023
DA - 2023/07/17
PB - OOO Zhurnal "Mendeleevskie Soobshcheniya"
SP - 448-450
IS - 4
VL - 33
SN - 0959-9436
SN - 1364-551X
ER -
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@article{2023_Elinson,
author = {M. N. Elinson and Anatoly N. Vereshchagin and Yuliya E. Ryzhkova and Kirill A Karpenko and Varvara M Kalashnikova and M. P. Egorov},
title = {An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold},
journal = {Mendeleev Communications},
year = {2023},
volume = {33},
publisher = {OOO Zhurnal "Mendeleevskie Soobshcheniya"},
month = {jul},
url = {https://doi.org/10.1016/j.mencom.2023.06.002},
number = {4},
pages = {448--450},
doi = {10.1016/j.mencom.2023.06.002}
}
MLA
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Elinson, M. N., et al. “An expedient cyclization of polyfunctional (aryl)(pyrimidinyl)(pyranyl)methanes into spiro[furo[3,2-c]pyran-2,5’-pyrimidine] scaffold.” Mendeleev Communications, vol. 33, no. 4, Jul. 2023, pp. 448-450. https://doi.org/10.1016/j.mencom.2023.06.002.