Open Access
COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis.
Тип публикации: Journal Article
Дата публикации: 2005-10-01
scimago Q1
wos Q1
БС1
SJR: 2.664
CiteScore: 18.6
Impact factor: 10.5
ISSN: 10436618, 10961186
PubMed ID:
15939622
Pharmacology
Краткое описание
We report on the inhibitory activity of the NSAIDs meloxicam, carprofen, phenylbutazone and flunixin, on blood cyclooxygenases in the horse using in vitro enzyme-linked assays. As expected, comparison of IC50 indicated that meloxicam and carprofen are more selective inhibitors of COX-2 than phenylbutazone and flunixin; meloxicam was the most advantageous for horses of four NSAIDs examined. However at IC80, phenylbutazone (+134.4%) and flunixin (+29.7%) had greater COX-2 selectivity than at IC50, and meloxicam (-41.2%) and carprofen (-12.9%) had lower COX-2 selectivity than at IC50. We therefore propose that the selectivity of NSAIDs should be assessed at the 80% as well as 50% inhibition level.
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Beretta C., Garavaglia G., Cavalli M. COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis. // Pharmacological Research. 2005. Vol. 52. No. 4. pp. 302-306.
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Beretta C., Garavaglia G., Cavalli M. COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis. // Pharmacological Research. 2005. Vol. 52. No. 4. pp. 302-306.
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TY - JOUR
DO - 10.1016/j.phrs.2005.04.004
UR - https://doi.org/10.1016/j.phrs.2005.04.004
TI - COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis.
T2 - Pharmacological Research
AU - Beretta, C.
AU - Garavaglia, G
AU - Cavalli, M.
PY - 2005
DA - 2005/10/01
PB - Elsevier
SP - 302-306
IS - 4
VL - 52
PMID - 15939622
SN - 1043-6618
SN - 1096-1186
ER -
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@article{2005_Beretta,
author = {C. Beretta and G Garavaglia and M. Cavalli},
title = {COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis.},
journal = {Pharmacological Research},
year = {2005},
volume = {52},
publisher = {Elsevier},
month = {oct},
url = {https://doi.org/10.1016/j.phrs.2005.04.004},
number = {4},
pages = {302--306},
doi = {10.1016/j.phrs.2005.04.004}
}
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Beretta, C., et al. “COX-1 and COX-2 inhibition in horse blood by phenylbutazone, flunixin, carprofen and meloxicam: an in vitro analysis..” Pharmacological Research, vol. 52, no. 4, Oct. 2005, pp. 302-306. https://doi.org/10.1016/j.phrs.2005.04.004.