Tetrahedron Letters

, том 51 , издание 48 , страницы 6325-6328

Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors

Тип публикации: Journal Article

Дата публикации: 2010-12-01

Elsevier

Tetrahedron Letters

scimago Q3

wos Q3

БС2

SJR: 0.334

CiteScore: 3.2

Impact factor: 1.5

ISSN: 00404039, 18733581

DOI: 10.1016/j.tetlet.2010.09.121

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Organic Chemistry

Drug Discovery

Biochemistry

Краткое описание

3-(Chloromethyl)coumarins, obtained via acid-catalysed cyclisation of salicylaldehyde-derived Baylis–Hillman adducts, have been treated with propargylamine; reaction of the resulting 3-alkynylmethylcoumarins with azidothymidine (AZT) in the presence of a Cu(I) catalyst has afforded a series of cycloaddition products for evaluation, in their own right, as potential dual-action HIV-1 protease and non-nucleoside reverse transcriptase inhibitors, and as scaffolds for further structural elaboration.

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Olomola T. O. et al. Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors // Tetrahedron Letters. 2010. Vol. 51. No. 48. pp. 6325-6328.

ГОСТ со всеми авторами (до 50) Скопировать

Olomola T. O., Klein R., Lobb K. A., Sayed Y., Kaye P. T. Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors // Tetrahedron Letters. 2010. Vol. 51. No. 48. pp. 6325-6328.

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TY - JOUR

DO - 10.1016/j.tetlet.2010.09.121

UR - https://doi.org/10.1016/j.tetlet.2010.09.121

TI - Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors

T2 - Tetrahedron Letters

AU - Olomola, Temitope O

AU - Klein, Rosalyn

AU - Lobb, Kevin Alan

AU - Sayed, Yasien

AU - Kaye, P. T.

PY - 2010

DA - 2010/12/01

PB - Elsevier

SP - 6325-6328

IS - 48

VL - 51

SN - 0040-4039

SN - 1873-3581

ER -

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@article{2010_Olomola,

author = {Temitope O Olomola and Rosalyn Klein and Kevin Alan Lobb and Yasien Sayed and P. T. Kaye},

title = {Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors},

journal = {Tetrahedron Letters},

year = {2010},

volume = {51},

publisher = {Elsevier},

month = {dec},

url = {https://doi.org/10.1016/j.tetlet.2010.09.121},

number = {48},

pages = {6325--6328},

doi = {10.1016/j.tetlet.2010.09.121}

}

MLA

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MLA Скопировать

Olomola, Temitope O., et al. “Towards the synthesis of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors.” Tetrahedron Letters, vol. 51, no. 48, Dec. 2010, pp. 6325-6328. https://doi.org/10.1016/j.tetlet.2010.09.121.

Издатель

Elsevier

Журнал

Tetrahedron Letters

scimago Q3

wos Q3

БС2

SJR

0.334

CiteScore

3.2

Impact factor

1.5

ISSN

00404039 (Print)

18733581 (Electronic)