Elsevier
Tetrahedron Letters
,  том 53 ,  издание 44 ,  страницы 5833-5836

Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist

Тип публикации: Journal Article
Дата публикации: 2012-10-01
Elsevier
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wos Q3
БС2
SJR: 0.334
CiteScore: 3.2
Impact factor: 1.5
ISSN: 00404039, 18733581
Organic Chemistry
Drug Discovery
Biochemistry
Краткое описание
The development of an efficient and scalable synthetic route to prepare the selective D2 partial agonist (1) is described here. Regioselective nitration of tetrahydrobenzazepine 2, followed by reductive amination, hydrogenation, and oxidative cyclization afforded 1 in good yield, without the need of column chromatography.
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Xiong H. et al. Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist // Tetrahedron Letters. 2012. Vol. 53. No. 44. pp. 5833-5836.
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Xiong H., Wu Y., Lehr S. G., BLACKWELL W., Steelman G., Hulsizer J., Urbanek R. A. Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist // Tetrahedron Letters. 2012. Vol. 53. No. 44. pp. 5833-5836.
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TY - JOUR
DO - 10.1016/j.tetlet.2012.08.035
UR - https://doi.org/10.1016/j.tetlet.2012.08.035
TI - Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist
T2 - Tetrahedron Letters
AU - Xiong, Hui
AU - Wu, Ye
AU - Lehr, Scott G
AU - BLACKWELL, WILLIAM
AU - Steelman, Gary
AU - Hulsizer, Jim
AU - Urbanek, Rebecca A.
PY - 2012
DA - 2012/10/01
PB - Elsevier
SP - 5833-5836
IS - 44
VL - 53
SN - 0040-4039
SN - 1873-3581
ER -
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@article{2012_Xiong,
author = {Hui Xiong and Ye Wu and Scott G Lehr and WILLIAM BLACKWELL and Gary Steelman and Jim Hulsizer and Rebecca A. Urbanek},
title = {Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist},
journal = {Tetrahedron Letters},
year = {2012},
volume = {53},
publisher = {Elsevier},
month = {oct},
url = {https://doi.org/10.1016/j.tetlet.2012.08.035},
number = {44},
pages = {5833--5836},
doi = {10.1016/j.tetlet.2012.08.035}
}
MLA
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Xiong, Hui, et al. “Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist.” Tetrahedron Letters, vol. 53, no. 44, Oct. 2012, pp. 5833-5836. https://doi.org/10.1016/j.tetlet.2012.08.035.