Monoamine transporter pharmacology and mutant mice
Тип публикации: Journal Article
Дата публикации: 2002-08-01
scimago Q1
wos Q1
БС1
SJR: 3.771
CiteScore: 25.7
Impact factor: 19.9
ISSN: 01656147, 18733735
PubMed ID:
12377578
Pharmacology
Toxicology
Краткое описание
Monoamine transporters, such as the dopamine transporter, 5-HT transporter and noradrenaline transporter, in the plasma membrane provide effective control over the intensity of monoamine-mediated signaling by recapturing neurotransmitters released by presynaptic neurons. These proteins represent established targets for several psychotropic drugs, including psychostimulants and antidepressants; however, important issues regarding the selectivity and mechanisms of action of these drugs remain unresolved. Although monoamine transporter knockout mice have profound changes in neurotransmission, they provide useful in vivo models to analyze the effects of psychotropic drugs. In this review, we summarize recent insights into the pharmacology of psychotropic drugs using mice in which the genes encoding these transporters have been deleted.
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Gainetdinov R. R., Sotnikova T. D., Caron M. G. Monoamine transporter pharmacology and mutant mice // Trends in Pharmacological Sciences. 2002. Vol. 23. No. 8. pp. 367-373.
ГОСТ со всеми авторами (до 50)
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Gainetdinov R. R., Sotnikova T. D., Caron M. G. Monoamine transporter pharmacology and mutant mice // Trends in Pharmacological Sciences. 2002. Vol. 23. No. 8. pp. 367-373.
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TY - JOUR
DO - 10.1016/S0165-6147(02)02044-8
UR - https://doi.org/10.1016/S0165-6147(02)02044-8
TI - Monoamine transporter pharmacology and mutant mice
T2 - Trends in Pharmacological Sciences
AU - Gainetdinov, R. R.
AU - Sotnikova, Tatyana D.
AU - Caron, Marc G.
PY - 2002
DA - 2002/08/01
PB - Elsevier
SP - 367-373
IS - 8
VL - 23
PMID - 12377578
SN - 0165-6147
SN - 1873-3735
ER -
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@article{2002_Gainetdinov,
author = {R. R. Gainetdinov and Tatyana D. Sotnikova and Marc G. Caron},
title = {Monoamine transporter pharmacology and mutant mice},
journal = {Trends in Pharmacological Sciences},
year = {2002},
volume = {23},
publisher = {Elsevier},
month = {aug},
url = {https://doi.org/10.1016/S0165-6147(02)02044-8},
number = {8},
pages = {367--373},
doi = {10.1016/S0165-6147(02)02044-8}
}
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MLA
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Gainetdinov, R. R., et al. “Monoamine transporter pharmacology and mutant mice.” Trends in Pharmacological Sciences, vol. 23, no. 8, Aug. 2002, pp. 367-373. https://doi.org/10.1016/S0165-6147(02)02044-8.
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