volume 23 issue 15 pages 5804-5808

Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates

Publication typeJournal Article
Publication date2021-07-19
scimago Q1
wos Q1
SJR1.235
CiteScore8.7
Impact factor5.0
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract
The first asymmetric trifluoromethylated allylic alkylation of pyrazolones using α-(trifluoromethyl)alkenyl acetates as a novel trifluoromethylated allylation reagent is described, affording various functionalized chiral pyrazolones containing a trifluoromethylated allyl substituent in high yields with excellent regio-/enantio-/diastereoselectivities. Mechanistically, the double-bond migration of α-(trifluoromethyl)alkenyl acetates in the presence of 1,8-diazabicyclo[5.4.0]undec-7-ene is initial and interesting step. More importantly, this study is of significance in providing a novel and widely applicable trifluoromethyl-containing allylation reagent.
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GOST |
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GOST Copy
Li D. et al. Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates // Organic Letters. 2021. Vol. 23. No. 15. pp. 5804-5808.
GOST all authors (up to 50) Copy
Li D., Zhang W., Zhang S., Sun W., Zhao J., Wang B., Qu J., Zhou Y. Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates // Organic Letters. 2021. Vol. 23. No. 15. pp. 5804-5808.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1021/acs.orglett.1c01957
UR - https://doi.org/10.1021/acs.orglett.1c01957
TI - Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates
T2 - Organic Letters
AU - Li, Dong
AU - Zhang, Wande
AU - Zhang, Shuaibo
AU - Sun, Wuding
AU - Zhao, Jinfeng
AU - Wang, Baomin
AU - Qu, Jingping
AU - Zhou, Yuhan
PY - 2021
DA - 2021/07/19
PB - American Chemical Society (ACS)
SP - 5804-5808
IS - 15
VL - 23
PMID - 34279113
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2021_Li,
author = {Dong Li and Wande Zhang and Shuaibo Zhang and Wuding Sun and Jinfeng Zhao and Baomin Wang and Jingping Qu and Yuhan Zhou},
title = {Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates},
journal = {Organic Letters},
year = {2021},
volume = {23},
publisher = {American Chemical Society (ACS)},
month = {jul},
url = {https://doi.org/10.1021/acs.orglett.1c01957},
number = {15},
pages = {5804--5808},
doi = {10.1021/acs.orglett.1c01957}
}
MLA
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MLA Copy
Li, Dong, et al. “Palladium-Catalyzed Asymmetric Trifluoromethylated Allylic Alkylation of Pyrazolones Enabled by α-(Trifluoromethyl)alkenyl Acetates.” Organic Letters, vol. 23, no. 15, Jul. 2021, pp. 5804-5808. https://doi.org/10.1021/acs.orglett.1c01957.