том 18 издание 21 страницы 5748-5751

Synthesis of Chiral Azabicycles from Pyroglutaminols

Тип публикацииJournal Article
Дата публикации2016-10-27
scimago Q1
wos Q1
БС1
SJR1.235
CiteScore8.7
Impact factor5.0
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
The stereocontrolled synthesis of a range of substituted bicyclic morpholine and piperazine derivatives is reported from substituted pyroglutaminols via an intramolecular SN2 cyclization as the key step. This enantiospecific approach toward chiral bicyclic morpholines and piperazines offers new opportunities to access these challenging ring systems, which are becoming increasingly common motifs in drug discovery.
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Organic Process Research and Development
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Organic Letters
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Acta Crystallographica Section E: Crystallographic Communications
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European Journal of Organic Chemistry
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Wiley
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ГОСТ |
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Choi C. et al. Synthesis of Chiral Azabicycles from Pyroglutaminols // Organic Letters. 2016. Vol. 18. No. 21. pp. 5748-5751.
ГОСТ со всеми авторами (до 50) Скопировать
Choi C., Nuhant P., Mousseau J. J., Yang X., Gerstenberger B. S., Williams J. M., Wright S. W. Synthesis of Chiral Azabicycles from Pyroglutaminols // Organic Letters. 2016. Vol. 18. No. 21. pp. 5748-5751.
RIS |
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TY - JOUR
DO - 10.1021/acs.orglett.6b03024
UR - https://doi.org/10.1021/acs.orglett.6b03024
TI - Synthesis of Chiral Azabicycles from Pyroglutaminols
T2 - Organic Letters
AU - Choi, Chulho
AU - Nuhant, Philippe
AU - Mousseau, James J.
AU - Yang, Xiaojing
AU - Gerstenberger, Brian S
AU - Williams, Jessica M.
AU - Wright, Stephen W
PY - 2016
DA - 2016/10/27
PB - American Chemical Society (ACS)
SP - 5748-5751
IS - 21
VL - 18
PMID - 27786487
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2016_Choi,
author = {Chulho Choi and Philippe Nuhant and James J. Mousseau and Xiaojing Yang and Brian S Gerstenberger and Jessica M. Williams and Stephen W Wright},
title = {Synthesis of Chiral Azabicycles from Pyroglutaminols},
journal = {Organic Letters},
year = {2016},
volume = {18},
publisher = {American Chemical Society (ACS)},
month = {oct},
url = {https://doi.org/10.1021/acs.orglett.6b03024},
number = {21},
pages = {5748--5751},
doi = {10.1021/acs.orglett.6b03024}
}
MLA
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Choi, Chulho, et al. “Synthesis of Chiral Azabicycles from Pyroglutaminols.” Organic Letters, vol. 18, no. 21, Oct. 2016, pp. 5748-5751. https://doi.org/10.1021/acs.orglett.6b03024.