Recent Progress in Histone Demethylase Inhibitors
Тип публикации: Journal Article
Дата публикации: 2016-02-02
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR: 1.726
CiteScore: 11.5
Impact factor: 6.8
ISSN: 00222623, 15204804
PubMed ID:
26710088
Drug Discovery
Molecular Medicine
Краткое описание
There is increasing interest in targeting histone N-methyl-lysine demethylases (KDMs) with small molecules both for the generation of probes for target exploration and for therapeutic purposes. Here we update on previous reviews on the inhibition of the lysine-specific demethylases (LSDs or KDM1s) and JmjC families of N-methyl-lysine demethylases (JmjC KDMs, KDM2-7), focusing on the academic and patent literature from 2014 to date. We also highlight recent biochemical, biological, and structural studies which are relevant to KDM inhibitor development.
Найдено
Ничего не найдено, попробуйте изменить настройки фильтра.
Для доступа к списку цитирований публикации необходимо авторизоваться.
Для доступа к списку профилей, цитирующих публикацию, необходимо авторизоваться.
Топ-30
Журналы
|
2
4
6
8
10
|
|
|
European Journal of Medicinal Chemistry
10 публикаций, 5.75%
|
|
|
Journal of Medicinal Chemistry
9 публикаций, 5.17%
|
|
|
Bioorganic and Medicinal Chemistry Letters
8 публикаций, 4.6%
|
|
|
Bioorganic and Medicinal Chemistry
7 публикаций, 4.02%
|
|
|
bioRxiv
4 публикации, 2.3%
|
|
|
Molecules
3 публикации, 1.72%
|
|
|
Cancers
3 публикации, 1.72%
|
|
|
Nature Communications
3 публикации, 1.72%
|
|
|
Bioorganic Chemistry
3 публикации, 1.72%
|
|
|
Cell Chemical Biology
3 публикации, 1.72%
|
|
|
ChemMedChem
3 публикации, 1.72%
|
|
|
Angewandte Chemie
3 публикации, 1.72%
|
|
|
Angewandte Chemie - International Edition
3 публикации, 1.72%
|
|
|
ACS Medicinal Chemistry Letters
3 публикации, 1.72%
|
|
|
Chemical Reviews
3 публикации, 1.72%
|
|
|
Lipophilicity in Drug Action and Toxicology
3 публикации, 1.72%
|
|
|
Current Medicinal Chemistry
2 публикации, 1.15%
|
|
|
Philosophical Transactions of the Royal Society B: Biological Sciences
2 публикации, 1.15%
|
|
|
Future Medicinal Chemistry
2 публикации, 1.15%
|
|
|
Frontiers in Cell and Developmental Biology
2 публикации, 1.15%
|
|
|
Journal of Molecular Graphics and Modelling
2 публикации, 1.15%
|
|
|
ChemBioChem
2 публикации, 1.15%
|
|
|
Medicinal Research Reviews
2 публикации, 1.15%
|
|
|
ACS Chemical Biology
2 публикации, 1.15%
|
|
|
RSC Advances
2 публикации, 1.15%
|
|
|
Topics in Medicinal Chemistry
2 публикации, 1.15%
|
|
|
Advances in Experimental Medicine and Biology
2 публикации, 1.15%
|
|
|
Current Topics in Medicinal Chemistry
1 публикация, 0.57%
|
|
|
Oncotarget
1 публикация, 0.57%
|
|
|
2
4
6
8
10
|
Издатели
|
10
20
30
40
50
60
|
|
|
Elsevier
58 публикаций, 33.33%
|
|
|
Wiley
28 публикаций, 16.09%
|
|
|
American Chemical Society (ACS)
20 публикаций, 11.49%
|
|
|
Springer Nature
18 публикаций, 10.34%
|
|
|
MDPI
10 публикаций, 5.75%
|
|
|
Taylor & Francis
6 публикаций, 3.45%
|
|
|
Royal Society of Chemistry (RSC)
5 публикаций, 2.87%
|
|
|
Frontiers Media S.A.
4 публикации, 2.3%
|
|
|
openRxiv
4 публикации, 2.3%
|
|
|
Bentham Science Publishers Ltd.
3 публикации, 1.72%
|
|
|
The Royal Society
2 публикации, 1.15%
|
|
|
Spandidos Publications
2 публикации, 1.15%
|
|
|
SAGE
2 публикации, 1.15%
|
|
|
Oxford University Press
2 публикации, 1.15%
|
|
|
Impact Journals
1 публикация, 0.57%
|
|
|
Ovid Technologies (Wolters Kluwer Health)
1 публикация, 0.57%
|
|
|
F1000 Research
1 публикация, 0.57%
|
|
|
American Association for the Advancement of Science (AAAS)
1 публикация, 0.57%
|
|
|
Korean Society of Cancer Prevention
1 публикация, 0.57%
|
|
|
Annual Reviews
1 публикация, 0.57%
|
|
|
OAE Publishing Inc.
1 публикация, 0.57%
|
|
|
IMR Press
1 публикация, 0.57%
|
|
|
Autonomous Non-profit Organization Editorial Board of the journal Uspekhi Khimii
1 публикация, 0.57%
|
|
|
10
20
30
40
50
60
|
- Мы не учитываем публикации, у которых нет DOI.
- Статистика публикаций обновляется еженедельно.
Вы ученый?
Создайте профиль, чтобы получать персональные рекомендации коллег, конференций и новых статей.
Войти с ORCID
Метрики
174
Всего цитирований:
174
Цитирований c 2025:
10
(5.74%)
Цитировать
ГОСТ |
RIS |
BibTex |
MLA
Цитировать
ГОСТ
Скопировать
McAllister T. et al. Recent Progress in Histone Demethylase Inhibitors // Journal of Medicinal Chemistry. 2016. Vol. 59. No. 4. pp. 1308-1329.
ГОСТ со всеми авторами (до 50)
Скопировать
McAllister T., England K. S., Hopkinson R. J., Brennan P. M., Kawamura A., Schofield C. J. Recent Progress in Histone Demethylase Inhibitors // Journal of Medicinal Chemistry. 2016. Vol. 59. No. 4. pp. 1308-1329.
Цитировать
RIS
Скопировать
TY - JOUR
DO - 10.1021/acs.jmedchem.5b01758
UR - https://doi.org/10.1021/acs.jmedchem.5b01758
TI - Recent Progress in Histone Demethylase Inhibitors
T2 - Journal of Medicinal Chemistry
AU - McAllister, Tom
AU - England, Katherine S
AU - Hopkinson, Richard J.
AU - Brennan, Paul M.
AU - Kawamura, Akane
AU - Schofield, Christopher J.
PY - 2016
DA - 2016/02/02
PB - American Chemical Society (ACS)
SP - 1308-1329
IS - 4
VL - 59
PMID - 26710088
SN - 0022-2623
SN - 1520-4804
ER -
Цитировать
BibTex (до 50 авторов)
Скопировать
@article{2016_McAllister,
author = {Tom McAllister and Katherine S England and Richard J. Hopkinson and Paul M. Brennan and Akane Kawamura and Christopher J. Schofield},
title = {Recent Progress in Histone Demethylase Inhibitors},
journal = {Journal of Medicinal Chemistry},
year = {2016},
volume = {59},
publisher = {American Chemical Society (ACS)},
month = {feb},
url = {https://doi.org/10.1021/acs.jmedchem.5b01758},
number = {4},
pages = {1308--1329},
doi = {10.1021/acs.jmedchem.5b01758}
}
Цитировать
MLA
Скопировать
McAllister, Tom, et al. “Recent Progress in Histone Demethylase Inhibitors.” Journal of Medicinal Chemistry, vol. 59, no. 4, Feb. 2016, pp. 1308-1329. https://doi.org/10.1021/acs.jmedchem.5b01758.
Ошибка в публикации?