том 85 издание 12 страницы 8149-8156

Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction

Тип публикацииJournal Article
Дата публикации2020-05-22
SCImago Q2
WOS Q1
БС1
SJR0.604
CiteScore6.1
Impact factor3.6
ISSN00223263, 15206904
Organic Chemistry
Краткое описание
The total synthesis of iheyamine A from readily available ethyl 2-aminocinnamate and 5-methoxyindole-2-carboxaldehyde is described. The cyanide-catalyzed imino-Stetter reaction of an aldimine derived from ethyl 2-aminocinnamate and 5-methoxyindole-2-carboxaldehyde provided the desired unsymmetrical 2,2'-bisindole-3-acetic acid derivative. The subsequent introduction of an amino group at the C-3' position, followed by the formation of the azepine ring, completed the total synthesis of iheyamine A.
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ГОСТ |
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Jeon J., Kim H. J., Cheon C. H. Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction // Journal of Organic Chemistry. 2020. Vol. 85. No. 12. pp. 8149-8156.
ГОСТ со всеми авторами (до 50) Скопировать
Jeon J., Kim H. J., Cheon C. H. Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction // Journal of Organic Chemistry. 2020. Vol. 85. No. 12. pp. 8149-8156.
RIS |
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TY - JOUR
DO - 10.1021/acs.joc.0c01051
UR - https://doi.org/10.1021/acs.joc.0c01051
TI - Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction
T2 - Journal of Organic Chemistry
AU - Jeon, Jiye
AU - Kim, Hyung Joo
AU - Cheon, Cheol Hong
PY - 2020
DA - 2020/05/22
PB - American Chemical Society (ACS)
SP - 8149-8156
IS - 12
VL - 85
PMID - 32441099
SN - 0022-3263
SN - 1520-6904
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2020_Jeon,
author = {Jiye Jeon and Hyung Joo Kim and Cheol Hong Cheon},
title = {Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction},
journal = {Journal of Organic Chemistry},
year = {2020},
volume = {85},
publisher = {American Chemical Society (ACS)},
month = {may},
url = {https://doi.org/10.1021/acs.joc.0c01051},
number = {12},
pages = {8149--8156},
doi = {10.1021/acs.joc.0c01051}
}
MLA
Цитировать
Jeon, Jiye, et al. “Total Synthesis of Iheyamine A via the Cyanide-Catalyzed Imino-Stetter Reaction.” Journal of Organic Chemistry, vol. 85, no. 12, May. 2020, pp. 8149-8156. https://doi.org/10.1021/acs.joc.0c01051.
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