том 24 издание 32 страницы 6066-6071

N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling

Тип публикацииJournal Article
Дата публикации2022-08-05
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR1.007
CiteScore7.7
Impact factor4.7
ISSN15237060, 15237052
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Краткое описание
N-Heterocyclic carbene (NHC)-catalyzed umpolung of cyclopent-4-ene-1,3-diones that proceeds via the generation of nucleophilic deoxy-Breslow intermediates is presented. The carbene generated from a commercially available thiazolium salt catalyzed the cross-coupling between cyclopent-4-ene-1,3-diones and isatins to furnish the functionalized oxindoles in moderate to good yields with good functional group compatibility. The key deoxy-Breslow intermediates were isolated and characterized by X-ray analysis. Detailed mechanistic studies are also presented.
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ГОСТ |
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Barik S., Shee S., Biju A. N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling // Organic Letters. 2022. Vol. 24. No. 32. pp. 6066-6071.
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Barik S., Shee S., Biju A. N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling // Organic Letters. 2022. Vol. 24. No. 32. pp. 6066-6071.
RIS |
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TY - JOUR
DO - 10.1021/acs.orglett.2c02413
UR - https://doi.org/10.1021/acs.orglett.2c02413
TI - N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling
T2 - Organic Letters
AU - Barik, Shilpa
AU - Shee, Sayan
AU - Biju, A.T
PY - 2022
DA - 2022/08/05
PB - American Chemical Society (ACS)
SP - 6066-6071
IS - 32
VL - 24
PMID - 35930323
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
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@article{2022_Barik,
author = {Shilpa Barik and Sayan Shee and A.T Biju},
title = {N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling},
journal = {Organic Letters},
year = {2022},
volume = {24},
publisher = {American Chemical Society (ACS)},
month = {aug},
url = {https://doi.org/10.1021/acs.orglett.2c02413},
number = {32},
pages = {6066--6071},
doi = {10.1021/acs.orglett.2c02413}
}
MLA
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Barik, Shilpa, et al. “N-Heterocyclic Carbene-Catalyzed Umpolung of Cyclopent-4-ene-1,3-diones for Activated Olefin–Isatin Cross-Coupling.” Organic Letters, vol. 24, no. 32, Aug. 2022, pp. 6066-6071. https://doi.org/10.1021/acs.orglett.2c02413.
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