Open Access
Open access
American Chemical Society (ACS)
ACS Omega
,  volume 5 ,  issue 25 ,  pages 15681-15690

Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation

Publication type: Journal Article
Publication date: 2020-06-18
American Chemical Society (ACS)
scimago Q1
wos Q2
SJR: 0.773
CiteScore: 7.1
Impact factor: 4.3
ISSN: 24701343
General Chemistry
General Chemical Engineering
Abstract
A convenient approach to [1,2,5]oxadiazolo[3′,4′:5,6]pyrazino[2,3-b]indoles and their heteroannulated analogues bearing various aryl substituents in the backbone has been developed. This synthetic protocol is based on Pd-catalyzed Buchwald–Hartwig and subsequent annulation by intramolecular oxidative cyclodehydrogenation. The photophysical properties for new polycycles have been measured.
Found 
Found 
2 citations
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GOST Copy
Kvashnin Y. A. et al. Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation // ACS Omega. 2020. Vol. 5. No. 25. pp. 15681-15690.
GOST all authors (up to 50) Copy
Kvashnin Y. A., Verbitskiy E. V., Zhilina E. F., Rusinov G. L., Chupakhin O. N., Charushin V. Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation // ACS Omega. 2020. Vol. 5. No. 25. pp. 15681-15690.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1021/acsomega.0c01945
UR - https://doi.org/10.1021/acsomega.0c01945
TI - Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation
T2 - ACS Omega
AU - Kvashnin, Yuriy A
AU - Verbitskiy, Egor V
AU - Zhilina, Ekaterina F.
AU - Rusinov, Gennady L.
AU - Chupakhin, O. N.
AU - Charushin, Valery
PY - 2020
DA - 2020/06/18
PB - American Chemical Society (ACS)
SP - 15681-15690
IS - 25
VL - 5
PMID - 32637843
SN - 2470-1343
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2020_Kvashnin,
author = {Yuriy A Kvashnin and Egor V Verbitskiy and Ekaterina F. Zhilina and Gennady L. Rusinov and O. N. Chupakhin and Valery Charushin},
title = {Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation},
journal = {ACS Omega},
year = {2020},
volume = {5},
publisher = {American Chemical Society (ACS)},
month = {jun},
url = {https://doi.org/10.1021/acsomega.0c01945},
number = {25},
pages = {15681--15690},
doi = {10.1021/acsomega.0c01945}
}
MLA
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MLA Copy
Kvashnin, Yuriy A., et al. “Synthesis of Heteroannulated Indolopyrazines through Domino N–H Palladium-Catalyzed/Metal-Free Oxidative C–H Bond Activation.” ACS Omega, vol. 5, no. 25, Jun. 2020, pp. 15681-15690. https://doi.org/10.1021/acsomega.0c01945.