том 15 издание 7 страницы 331-334

Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis

Тип публикацииJournal Article
Дата публикации2013-06-06
БС1
SJR0.833
CiteScore
Impact factor3.9
ISSN21568952, 21568944
General Chemistry
General Medicine
Краткое описание
An efficient, standard, mild, and copper-free imidazole-1-sulfonyl azide hydrochloride-based diazo-transfer method was implemented in a set of four resins that cover a broad range of hydrophobicity. The imidazole-1-sulfonyl azide hydrochloride is easily prepared/commercially available, stable upon storage at 4 °C, and proved to be a suitable alternative to triflyl azide for diazo-transfer reactions in amine functionalized resins. We have successfully applied the azido resins for the conjugation of a TFA-labile Wang-type linker using Click Chemistry.
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ГОСТ |
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Castro V. et al. Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis // ACS Combinatorial Science. 2013. Vol. 15. No. 7. pp. 331-334.
ГОСТ со всеми авторами (до 50) Скопировать
Castro V., Blanco Canosa J. B., Rodrı́guez H., Albericio F. Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis // ACS Combinatorial Science. 2013. Vol. 15. No. 7. pp. 331-334.
RIS |
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TY - JOUR
DO - 10.1021/co4000437
UR - https://doi.org/10.1021/co4000437
TI - Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis
T2 - ACS Combinatorial Science
AU - Castro, Vida
AU - Blanco Canosa, Juan B
AU - Rodrı́guez, H.Ricardo
AU - Albericio, Fernando
PY - 2013
DA - 2013/06/06
PB - American Chemical Society (ACS)
SP - 331-334
IS - 7
VL - 15
PMID - 23721561
SN - 2156-8952
SN - 2156-8944
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2013_Castro,
author = {Vida Castro and Juan B Blanco Canosa and H.Ricardo Rodrı́guez and Fernando Albericio},
title = {Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis},
journal = {ACS Combinatorial Science},
year = {2013},
volume = {15},
publisher = {American Chemical Society (ACS)},
month = {jun},
url = {https://doi.org/10.1021/co4000437},
number = {7},
pages = {331--334},
doi = {10.1021/co4000437}
}
MLA
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Castro, Vida, et al. “Imidazole-1-sulfonyl Azide-Based Diazo-Transfer Reaction for the Preparation of Azido Solid Supports for Solid-Phase Synthesis.” ACS Combinatorial Science, vol. 15, no. 7, Jun. 2013, pp. 331-334. https://doi.org/10.1021/co4000437.
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