том 37 издание 25 страницы 4412-4416

Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation

Тип публикацииJournal Article
Дата публикации1994-12-01
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR1.726
CiteScore11.1
Impact factor7.3
ISSN00222623, 15204804
Drug Discovery
Molecular Medicine
Краткое описание
4-Phenyl-3-furoxancarbonitrile (2) affords nitric oxide under the action of thiol cofactors. Two principal products were isolated in the reaction with thiophenol: the phenylcyanoglyoxime (6) and 5-amino-3-phenyl-4-(phenylthio)isoxazole (7). Mechanisms which could account for the formation of these two products are discussed. Compound 2 is an efficient activator of the rat lung soluble guanylate cyclase, displays high vasodilatory activity on strips of rat thoracic aorta precontracted with noradrenaline, and is a potent inhibitor of platelet aggregation.
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ГОСТ |
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Medana C. et al. Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation // Journal of Medicinal Chemistry. 1994. Vol. 37. No. 25. pp. 4412-4416.
ГОСТ со всеми авторами (до 50) Скопировать
Medana C. Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation // Journal of Medicinal Chemistry. 1994. Vol. 37. No. 25. pp. 4412-4416.
RIS |
Цитировать
TY - JOUR
DO - 10.1021/jm00051a020
UR - https://doi.org/10.1021/jm00051a020
TI - Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation
T2 - Journal of Medicinal Chemistry
AU - Medana, Claudio
PY - 1994
DA - 1994/12/01
PB - American Chemical Society (ACS)
SP - 4412-4416
IS - 25
VL - 37
PMID - 7996554
SN - 0022-2623
SN - 1520-4804
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{1994_Medana,
author = {Claudio Medana},
title = {Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation},
journal = {Journal of Medicinal Chemistry},
year = {1994},
volume = {37},
publisher = {American Chemical Society (ACS)},
month = {dec},
url = {https://doi.org/10.1021/jm00051a020},
number = {25},
pages = {4412--4416},
doi = {10.1021/jm00051a020}
}
MLA
Цитировать
Medana, Claudio, et al. “Furoxans as Nitric Oxide Donors. 4-Phenyl-3-furoxancarbonitrile: Thiol-Mediated Nitric Oxide Release and Biological Evaluation.” Journal of Medicinal Chemistry, vol. 37, no. 25, Dec. 1994, pp. 4412-4416. https://doi.org/10.1021/jm00051a020.
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