Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands
Тип публикации: Journal Article
Дата публикации: 2003-07-18
scimago Q1
wos Q1
БС1
SJR: 1.801
CiteScore: 11.5
Impact factor: 6.8
ISSN: 00222623, 15204804
PubMed ID:
12904061
Drug Discovery
Molecular Medicine
Краткое описание
The structure-activity relationship studies on 2-quinolinecarboxamide peripheral benzodiazepine receptor (PBR) ligands have been refined with the aim of using these ligands as carriers of radionuclides and boron atoms. Some new ligands show enhanced affinity and steroidogenic activity with respect to reference compound 1 and are interesting candidates for radiolabeling and PET studies. Moreover, carborane derivative 3q, representing the first example of PBR ligand bearing a carborane cage, can be useful to explore an alternative mechanism in BNCT.
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ГОСТ
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Cappelli A. et al. Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands // Journal of Medicinal Chemistry. 2003. Vol. 46. No. 17. pp. 3568-3571.
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Cappelli A., Pericot Mohr G. L., Gallelli A., Giuliani G., Anzini M., Vomero S., Fresta M., Porcu P., MACIOCCO E., Concas A., Biggio G., Donati A. Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands // Journal of Medicinal Chemistry. 2003. Vol. 46. No. 17. pp. 3568-3571.
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TY - JOUR
DO - 10.1021/jm034068b
UR - https://doi.org/10.1021/jm034068b
TI - Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands
T2 - Journal of Medicinal Chemistry
AU - Cappelli, A.
AU - Pericot Mohr, Gal La
AU - Gallelli, Andrea
AU - Giuliani, Germano
AU - Anzini, Maurizio
AU - Vomero, Salvatore
AU - Fresta, Massimo
AU - Porcu, P.
AU - MACIOCCO, E.
AU - Concas, Alessandra
AU - Biggio, G.
AU - Donati, Alessandro
PY - 2003
DA - 2003/07/18
PB - American Chemical Society (ACS)
SP - 3568-3571
IS - 17
VL - 46
PMID - 12904061
SN - 0022-2623
SN - 1520-4804
ER -
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@article{2003_Cappelli,
author = {A. Cappelli and Gal La Pericot Mohr and Andrea Gallelli and Germano Giuliani and Maurizio Anzini and Salvatore Vomero and Massimo Fresta and P. Porcu and E. MACIOCCO and Alessandra Concas and G. Biggio and Alessandro Donati},
title = {Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands},
journal = {Journal of Medicinal Chemistry},
year = {2003},
volume = {46},
publisher = {American Chemical Society (ACS)},
month = {jul},
url = {https://doi.org/10.1021/jm034068b},
number = {17},
pages = {3568--3571},
doi = {10.1021/jm034068b}
}
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MLA
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Cappelli, A., et al. “Structure−Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands.” Journal of Medicinal Chemistry, vol. 46, no. 17, Jul. 2003, pp. 3568-3571. https://doi.org/10.1021/jm034068b.