Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases
Тип публикации: Journal Article
Дата публикации: 2008-10-23
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR: 1.726
CiteScore: 11.5
Impact factor: 6.8
ISSN: 00222623, 15204804
PubMed ID:
18942826
Drug Discovery
Molecular Medicine
Краткое описание
The dynamic methylation of histone lysyl residues plays an important role in biology by regulating transcription, maintaining genomic integrity, and by contributing to epigenetic effects. Here we describe a variety of inhibitor scaffolds that inhibit the human 2-oxoglutarate-dependent JMJD2 subfamily of histone demethylases. Combined with structural data, these chemical starting points will be useful to generate small-molecule probes to analyze the physiological roles of these enzymes in epigenetic signaling.
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ГОСТ
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Rose N. R. et al. Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases // Journal of Medicinal Chemistry. 2008. Vol. 51. No. 22. pp. 7053-7056.
ГОСТ со всеми авторами (до 50)
Скопировать
Rose N. R., Ng S. S., Mecinović J., Liénard B. M. R., Bello S. H., Sun Z., McDonough M., Oppermann U. C., Schofield C. J. Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases // Journal of Medicinal Chemistry. 2008. Vol. 51. No. 22. pp. 7053-7056.
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RIS
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TY - JOUR
DO - 10.1021/jm800936s
UR - https://doi.org/10.1021/jm800936s
TI - Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases
T2 - Journal of Medicinal Chemistry
AU - Rose, Nathan R
AU - Ng, Stanley S
AU - Mecinović, Jasmin
AU - Liénard, Benoît M R
AU - Bello, Simon H
AU - Sun, Zhe
AU - McDonough, Michael
AU - Oppermann, Udo C.I.
AU - Schofield, Christopher J.
PY - 2008
DA - 2008/10/23
PB - American Chemical Society (ACS)
SP - 7053-7056
IS - 22
VL - 51
PMID - 18942826
SN - 0022-2623
SN - 1520-4804
ER -
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@article{2008_Rose,
author = {Nathan R Rose and Stanley S Ng and Jasmin Mecinović and Benoît M R Liénard and Simon H Bello and Zhe Sun and Michael McDonough and Udo C.I. Oppermann and Christopher J. Schofield},
title = {Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases},
journal = {Journal of Medicinal Chemistry},
year = {2008},
volume = {51},
publisher = {American Chemical Society (ACS)},
month = {oct},
url = {https://doi.org/10.1021/jm800936s},
number = {22},
pages = {7053--7056},
doi = {10.1021/jm800936s}
}
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MLA
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Rose, Nathan R., et al. “Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases.” Journal of Medicinal Chemistry, vol. 51, no. 22, Oct. 2008, pp. 7053-7056. https://doi.org/10.1021/jm800936s.
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