Hydrogel Nanoparticles with Thermally Controlled Drug Release
Тип публикации: Journal Article
Дата публикации: 2014-06-12
scimago Q1
wos Q1
БС1
SJR: 1.287
CiteScore: 8.9
Impact factor: 5.2
ISSN: 21611653
PubMed ID:
25419487
Materials Chemistry
Organic Chemistry
Inorganic Chemistry
Polymers and Plastics
Краткое описание
Improving the therapeutic efficacy and reducing systemic side effects of drugs is an important aspect in chemotherapy. The strategy presented here is the use of cisplatin loaded, temperature-sensitive, hydrogel nanoparticles (CisPt-NPs) and their ability to deliver and release chemodrugs selectively, based on thermal stimuli. The specially synthesized CisPt-NPs show a temperature-dependent increase of cisplatin release, at neutral pH (as in blood and normal tissue), in both the presence and absence of common metallic ions, as well as at the low pH found in lysosomes, where endocytosed NPs often localize. These CisPt-NPs were uptaken by breast cancer MDA-MB-435 cells, via endocytosis, and then mostly localized in the lysosomes. The in vitro cytotoxicity tests show that these CisPt-NPs have a significantly better efficacy at the slightly elevated temperatures. Potential applications are discussed.
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ГОСТ
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Shirakura T. et al. Hydrogel Nanoparticles with Thermally Controlled Drug Release // ACS Macro Letters. 2014. Vol. 3. No. 7. pp. 602-606.
ГОСТ со всеми авторами (до 50)
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Shirakura T., Kelson T. J., Ray A., Malyarenko A. E., Kopelman R. Hydrogel Nanoparticles with Thermally Controlled Drug Release // ACS Macro Letters. 2014. Vol. 3. No. 7. pp. 602-606.
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RIS
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TY - JOUR
DO - 10.1021/mz500231e
UR - https://doi.org/10.1021/mz500231e
TI - Hydrogel Nanoparticles with Thermally Controlled Drug Release
T2 - ACS Macro Letters
AU - Shirakura, Teppei
AU - Kelson, Taylor J
AU - Ray, Aniruddha
AU - Malyarenko, Antonina E
AU - Kopelman, Raoul
PY - 2014
DA - 2014/06/12
PB - American Chemical Society (ACS)
SP - 602-606
IS - 7
VL - 3
PMID - 25419487
SN - 2161-1653
ER -
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BibTex (до 50 авторов)
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@article{2014_Shirakura,
author = {Teppei Shirakura and Taylor J Kelson and Aniruddha Ray and Antonina E Malyarenko and Raoul Kopelman},
title = {Hydrogel Nanoparticles with Thermally Controlled Drug Release},
journal = {ACS Macro Letters},
year = {2014},
volume = {3},
publisher = {American Chemical Society (ACS)},
month = {jun},
url = {https://doi.org/10.1021/mz500231e},
number = {7},
pages = {602--606},
doi = {10.1021/mz500231e}
}
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MLA
Скопировать
Shirakura, Teppei, et al. “Hydrogel Nanoparticles with Thermally Controlled Drug Release.” ACS Macro Letters, vol. 3, no. 7, Jun. 2014, pp. 602-606. https://doi.org/10.1021/mz500231e.