volume 12 issue 24 pages 5712-5715

Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides

Publication typeJournal Article
Publication date2010-12-17
scimago Q1
wos Q1
SJR1.235
CiteScore8.7
Impact factor5.0
ISSN15237060, 15237052
PubMed ID:  21086980
Organic Chemistry
Biochemistry
Physical and Theoretical Chemistry
Abstract
N-aryltriazole nucleosides are new chemical entities with potential biological activity. The two phosphor ligands, Synphos and Xantphos, had a selective and effective impact on Pd-catalyzed C-N coupling with the 5- and 3-bromotriazole acyclonucleoside isomers, affording the corresponding and otherwise difficult to achieve N-aryltriazole nucleosides with good to excellent yields. In addition, two of the synthesized nucleosides showed superior anticancer activity against drug-resistant pancreatic cancer, compared to the reference drug gemcitabine.
Found 

Top-30

Journals

1
Chemistry of Heterocyclic Compounds
1 publication, 7.14%
Scientific Reports
1 publication, 7.14%
Cancer Letters
1 publication, 7.14%
Ultrasonics Sonochemistry
1 publication, 7.14%
European Journal of Medicinal Chemistry
1 publication, 7.14%
Current Protocols
1 publication, 7.14%
Chemistry - A European Journal
1 publication, 7.14%
Journal of Medicinal Chemistry
1 publication, 7.14%
Inorganic Chemistry Frontiers
1 publication, 7.14%
New Journal of Chemistry
1 publication, 7.14%
Organic and Biomolecular Chemistry
1 publication, 7.14%
Mini-Reviews in Organic Chemistry
1 publication, 7.14%
Mendeleev Communications
1 publication, 7.14%
1

Publishers

1
2
3
4
Elsevier
4 publications, 28.57%
Royal Society of Chemistry (RSC)
3 publications, 21.43%
Springer Nature
2 publications, 14.29%
Wiley
2 publications, 14.29%
American Chemical Society (ACS)
1 publication, 7.14%
Bentham Science Publishers Ltd.
1 publication, 7.14%
OOO Zhurnal "Mendeleevskie Soobshcheniya"
1 publication, 7.14%
1
2
3
4
  • We do not take into account publications without a DOI.
  • Statistics recalculated weekly.

Are you a researcher?

Create a profile to get free access to personal recommendations for colleagues and new articles.
Metrics
14
Share
Cite this
GOST |
Cite this
GOST Copy
Fan Y. et al. Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides // Organic Letters. 2010. Vol. 12. No. 24. pp. 5712-5715.
GOST all authors (up to 50) Copy
Fan Y., Xia Y., Peng L. Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides // Organic Letters. 2010. Vol. 12. No. 24. pp. 5712-5715.
RIS |
Cite this
RIS Copy
TY - JOUR
DO - 10.1021/ol102537p
UR - https://doi.org/10.1021/ol102537p
TI - Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides
T2 - Organic Letters
AU - Fan, Yuting
AU - Xia, Yi
AU - Peng, Ling
PY - 2010
DA - 2010/12/17
PB - American Chemical Society (ACS)
SP - 5712-5715
IS - 24
VL - 12
PMID - 21086980
SN - 1523-7060
SN - 1523-7052
ER -
BibTex |
Cite this
BibTex (up to 50 authors) Copy
@article{2010_Fan,
author = {Yuting Fan and Yi Xia and Ling Peng},
title = {Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides},
journal = {Organic Letters},
year = {2010},
volume = {12},
publisher = {American Chemical Society (ACS)},
month = {dec},
url = {https://doi.org/10.1021/ol102537p},
number = {24},
pages = {5712--5715},
doi = {10.1021/ol102537p}
}
MLA
Cite this
MLA Copy
Fan, Yuting, et al. “Ligand-Mediated Highly Effective and Selective C−N Coupling for Synthesizing BioactiveN-Aryltriazole Acyclonucleosides.” Organic Letters, vol. 12, no. 24, Dec. 2010, pp. 5712-5715. https://doi.org/10.1021/ol102537p.