том 22 издание 10 страницы 3155-3161

Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes

Тип публикацииJournal Article
Дата публикации2020-04-21
SCImago Q1
Tоп 10% SCImago
WOS Q1
БС1
SJR1.811
CiteScore16
Impact factor10.6
ISSN14639262, 14639270
Environmental Chemistry
Pollution
Краткое описание
A nickel-based catalytic system for the regiospecific C2–H arylation of benzothiophene has been established. NiCl2(bpy) is used as a catalyst in combination with LiHMDS as a base in dioxane. The catalytic system is applicable to a variety of functionalized benzothiophenes, as well as other heteroarenes including thiophene, benzodithiophene, benzofuran and selenophene in combination with iodo aryl electrophiles. The role of LiHMDS as a uniquely potent base and a postulated mechanism are discussed. The applicability of this system is finally demonstrated for the synthesis of an intermediate of an active pharmaceutical ingredient.
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ГОСТ |
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Mohr Y. et al. Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes // Green Chemistry. 2020. Vol. 22. No. 10. pp. 3155-3161.
ГОСТ со всеми авторами (до 50) Скопировать
Mohr Y., Hisler G., Grousset L., Roux Y., Quadrelli E. A., Wisser F. M., Canivet J. Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes // Green Chemistry. 2020. Vol. 22. No. 10. pp. 3155-3161.
RIS |
Цитировать
TY - JOUR
DO - 10.1039/d0gc00917b
UR - https://xlink.rsc.org/?DOI=D0GC00917B
TI - Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes
T2 - Green Chemistry
AU - Mohr, Yorck
AU - Hisler, Gaëlle
AU - Grousset, Léonie
AU - Roux, Yoann
AU - Quadrelli, Elsje Alessandra
AU - Wisser, Florian M.
AU - Canivet, Jérôme
PY - 2020
DA - 2020/04/21
PB - Royal Society of Chemistry (RSC)
SP - 3155-3161
IS - 10
VL - 22
SN - 1463-9262
SN - 1463-9270
ER -
BibTex |
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BibTex (до 50 авторов) Скопировать
@article{2020_Mohr,
author = {Yorck Mohr and Gaëlle Hisler and Léonie Grousset and Yoann Roux and Elsje Alessandra Quadrelli and Florian M. Wisser and Jérôme Canivet},
title = {Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes},
journal = {Green Chemistry},
year = {2020},
volume = {22},
publisher = {Royal Society of Chemistry (RSC)},
month = {apr},
url = {https://xlink.rsc.org/?DOI=D0GC00917B},
number = {10},
pages = {3155--3161},
doi = {10.1039/d0gc00917b}
}
MLA
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Mohr, Yorck, et al. “Nickel-catalyzed and Li-mediated regiospecific C–H arylation of benzothiophenes.” Green Chemistry, vol. 22, no. 10, Apr. 2020, pp. 3155-3161. https://xlink.rsc.org/?DOI=D0GC00917B.
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